Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VDLPDIXFOKMSTE
|
7.3 | IC50 | 2 | — | |
VDUQDYKTCBRQHM
|
7.3 | IC50 | 2 | — | |
VEKYGTJVRVZEGI
|
7.3 | IC50 | 2 | — | |
VRBCYHMHHGOSNK
|
7.3 | IC50 | 2 | — | |
VUIDROACQSTZQH
|
7.3 | IC50 | 2 | — | |
VXZGPUGXEAWXNO
|
7.3 | IC50 | 2 | — | |
WDSAVECIVQHDAD
|
7.3 | IC50 | 3 | — | |
WDUZHMCHWHGCJJ
|
7.3 | IC50 | 2 | — | |
WEVPOLLVQNEHKK
|
7.3 | IC50 | 2 | — | |
WHCWRLSHTAKJAL
|
7.3 | IC50 | 2 | — | |
WQKACOSOCPWSJK
|
7.3 | IC50 | 2 | — | |
WZBKEVJKQOQNAH
|
7.3 | IC50 | 2 | — | |
XDXOWJKRCDMDIP
|
7.3 | IC50 | 3 | — | |
XELMNVUNDPFWPJ
|
7.3 | IC50 | 2 | — | |
XFRTYVGXWBPBFE
|
7.3 | IC50 | 2 | — | |
XHNADMLZYHEDEX
|
7.3 | IC50 | 2 | — | |
XPUMJVRQZHTBDO
|
7.3 | IC50 | 2 | — | |
XQAFICKHNGSCNA
|
7.3 | IC50 | 2 | — | |
XQLNJPZOTBTZON
|
7.3 | IC50 | 3 | — | |
XTRDBMQYGLGIDI
|
7.3 | IC50 | 2 | — | |
XUNRVYAOTKSKJA
|
7.3 | IC50 | 3 | — | |
YIKASSMFWGQONT
|
7.3 | IC50 | 2 | — | |
YOSQZDHYWPCOKE
|
7.3 | IC50 | 2 | — | |
YPLWWFWKQHTHLR
|
7.3 | IC50 | 2 | — | |
YTDZARLQOJJGAF
|
7.3 | IC50 | 2 | — | |
ZLBJRZPDABNGGW
|
7.3 | IC50 | 2 | — | |
ZNOGVOUAKUGQGF
|
7.3 | IC50 | 2 | — | |
ZOHCQNHQJRAISM
|
7.3 | IC50 | 2 | — | |
ZPGWQYUCSBEELY
|
7.3 | IC50 | 2 | — | |
ZQMDEILZYDIECZ
|
7.3 | IC50 | 2 | — | |
ZVGRBNITRNLZNZ
|
7.3 | IC50 | 2 | — | |
RENRJGXFTHYPPG
|
7.2 | IC50 | 2 | — | |
WDSAJBCCUSPKPI
|
7.2 | IC50 | 2 | — | |
CHGGBMTUUUUZHD
|
7.2 | IC50 | 2 | — | |
NKPYAWCAMKAQPM
|
7.2 | IC50 | 3 | — | |
MQZVKSLKRZNVIE
|
7.2 | IC50 | 2 | — | |
BYEDBMHYWDHELH
|
7.2 | IC50 | 2 | — | |
ISZNFBSZRWOLFS
|
7.2 | IC50 | 3 | — | |
ZBJQLGQZNRQUPU
|
7.2 | IC50 | 2 | — | |
HJCZOBLYJWGMDD
|
7.2 | IC50 | 2 | — | |
PEXUHARTKNIBDL
|
7.2 | IC50 | 2 | — | |
DVHKNGCCUGNVQZ
|
7.2 | IC50 | 2 | — | |
GKFUTHVAVQPTFA
|
7.2 | IC50 | 2 | — | |
ACRSYDLSAYZZOB
|
7.2 | IC50 | 2 | — | |
APAZLBBJADULHZ
|
7.2 | IC50 | 3 | — | |
ATJORKOQGVNLQY
|
7.2 | IC50 | 2 | — | |
BFLSJYFITVZAPW
|
7.2 | IC50 | 2 | — | |
CWVXEQPXRFPKEZ
|
7.2 | IC50 | 2 | — | |
FTBWNMAFKFLFHP
|
7.2 | IC50 | 2 | — | |
HOIBJSHJRQULFL
|
7.2 | IC50 | 3 | — |