Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
APYSBWNXLCWCMZ
|
7.3 | IC50 | 2 | — | |
AQUZXZFKJDBGDG
|
7.3 | IC50 | 2 | — | |
AQYBAGBDMKOZOT
|
7.3 | IC50 | 2 | — | |
AXNJSKMUFOXSLD
|
7.3 | IC50 | 2 | — | |
BONMFJRUCDDITM
|
7.3 | IC50 | 2 | — | |
BOQQQFJHHSQWBJ
|
7.3 | IC50 | 2 | — | |
BSKHIANLHIEMMY
|
7.3 | IC50 | 3 | — | |
BXIYCAYGWIHMHL
|
7.3 | IC50 | 2 | — | |
CDYZISGCDITLOI
|
7.3 | IC50 | 2 | — | |
CIJMJLPONKXFMU
|
7.3 | IC50 | 2 | — | |
CJEFTJNLWIVQJY
|
7.3 | IC50 | 2 | — | |
CLNZOVOBAXNFGG
|
7.3 | IC50 | 3 | — | |
CPRQKIQZMBAYGL
|
7.3 | IC50 | 3 | — | |
CQDXRRLRQTYPMT
|
7.3 | IC50 | 2 | — | |
CRAHFBSLWSAFHP
|
7.3 | IC50 | 3 | — | |
CXTQTURBDSEPDD
|
7.3 | IC50 | 2 | — | |
DGGBLEYOYXWXFD
|
7.3 | IC50 | 2 | — | |
DHHXPZKYXUDVQR
|
7.3 | IC50 | 2 | — | |
DLOQHHJANJFFJT
|
7.3 | IC50 | 2 | — | |
DNZFTJMJVDARQT
|
7.3 | IC50 | 2 | — | |
DQADWISJUULUAY
|
7.3 | IC50 | 2 | — | |
DRKPXDOCDDPDAI
|
7.3 | IC50 | 2 | — | |
DRNMVUQKFQVVHB
|
7.3 | IC50 | 2 | — | |
DUFQTWQYCOXKIC
|
7.3 | IC50 | 2 | — | |
DWHMPDFQOZEIQB
|
7.3 | IC50 | 2 | — | |
DXOOLCNUKDSRGP
|
7.3 | IC50 | 2 | — | |
DZGNYCKQISDLDR
|
7.3 | IC50 | 2 | — | |
FGNVSNWNINHOKH
|
7.3 | IC50 | 2 | — | |
FKEIYILKGUQVFR
|
7.3 | IC50 | 2 | — | |
FOIQFGDFWWNIAL
|
7.3 | IC50 | 2 | — | |
FQBQJUGLJKQFMK
|
7.3 | IC50 | 2 | — | |
FVDRXYMBNGVDPG
|
7.3 | IC50 | 2 | — | |
FWMSQWKYWWGJGB
|
7.3 | IC50 | 2 | — | |
GBGXUVPPNWEOLE
|
7.3 | IC50 | 3 | — | |
GECDPIJUZSAHIP
|
7.3 | IC50 | 2 | — | |
GOYIOFDJRGFRPE
|
7.3 | IC50 | 2 | — | |
GQROZXUHNBGXCR
|
7.3 | IC50 | 2 | — | |
GSMUZHMKXAHHFV
|
7.3 | IC50 | 2 | — | |
GTZDUBKNXPYACI
|
7.3 | IC50 | 2 | — | |
HFELIBJRXABNGD
|
7.3 | IC50 | 2 | — | |
HJUSYDIJANMTDQ
|
7.3 | IC50 | 2 | — | |
HLCJVZCFIIVFHT
|
7.3 | IC50 | 2 | — | |
HOFZBTJHUHUCHK
|
7.3 | IC50 | 2 | — | |
HUABRDTUMVFDGX
|
7.3 | IC50 | 2 | — | |
HWVDGRPNGIETSR
|
7.3 | IC50 | 2 | — | |
IGEOKPLPEDYNCW
|
7.3 | IC50 | 2 | — | |
IHHDUMSWPGIXPS
|
7.3 | IC50 | 2 | — | |
IICIPTUGFWJYHL
|
7.3 | IC50 | 2 | — | |
IXEXFVBVSLCJNA
|
7.3 | IC50 | 2 | — | |
IYCAKFOXGQBZQZ
|
7.3 | IC50 | 2 | — |