Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OPZZIKZUGSMEPY
|
7.4 | IC50 | 2 | — | |
PXNSUHQVXVDKFQ
|
7.4 | IC50 | 2 | — | |
RDKZTOQDJHEFQX
|
7.4 | IC50 | 2 | — | |
RXZOMMSIRRSXQW
|
7.4 | IC50 | 4 | — | |
ZYMMXVOIYKLHKH
|
7.4 | IC50 | 2 | — | |
APJOBTGOJXGDGH
|
7.4 | IC50 | 2 | — | |
AXMGRXURKXGCPI
|
7.4 | IC50 | 3 | — | |
CWRXCQQDEOGGAA
|
7.4 | IC50 | 2 | — | |
GZECANYKHKCEFF
|
7.4 | IC50 | 2 | — | |
LNNZWVZSBLLGRK
|
7.4 | IC50 | 2 | — | |
WRYYRMHEPCBQIZ
|
7.4 | IC50 | 2 | — | |
ZNGCWFPZUBLLOJ
|
7.4 | IC50 | 2 | — | |
GVZMDMVDKHKLPJ
|
7.4 | IC50 | 2 | — | |
KOZFSFOOLUUIGY
|
7.4 | Kd | 88 | Yes | |
NMQCDRLEHHKROH
|
7.4 | IC50 | 2 | — | |
DNINGYYWXPRQDJ
|
7.4 | Kd | 4 | — | |
FQIGYFHTRSLGKQ
|
7.4 | IC50 | 2 | — | |
VXGYSGCTPBOVEG
|
7.4 | IC50 | 3 | — | |
BCOMIOVRJUNIKO
|
7.4 | IC50 | 2 | — | |
DRUZOODDDHIXAI
|
7.4 | IC50 | 2 | — | |
HMNKBFFXICTTJO
|
7.4 | IC50 | 3 | — | |
WLCODBRLUVZHCP
|
7.3 | IC50 | 3 | — | |
CSTHTXUPJYUFSY
|
7.3 | IC50 | 2 | — | |
RHZIUVRWDZLXFG
|
7.3 | IC50 | 3 | — | |
VRGJIZUIODIMGX
|
7.3 | IC50 | 3 | — | |
ZOEILZXFYPPMTR
|
7.3 | IC50 | 2 | — | |
IDDANJDHVDUCCU
|
7.3 | IC50 | 2 | — | |
FFJXATKZPJXQMA
|
7.3 | IC50 | 2 | — | |
QNKFAXRCZUFWGQ
|
7.3 | IC50 | 3 | — | |
WQIPRNUEYVQWKW
|
7.3 | IC50 | 2 | — | |
BGQOUQWQPRPBKN
|
7.3 | IC50 | 7 | — | |
GJZCXJLZZFATOM
|
7.3 | IC50 | 2 | — | |
XBBFRFFVOXSJOR
|
7.3 | IC50 | 2 | — | |
XBVQPBVYQLZBGU
|
7.3 | IC50 | 2 | — | |
XSIQDWROCVFQSV
|
7.3 | IC50 | 2 | — | |
FPYULJCYPOLXGV
|
7.3 | IC50 | 2 | — | |
RWUOCYNYQYDGGU
|
7.3 | IC50 | 2 | — | |
FUKYTTWUNYCSJG
|
7.3 | IC50 | 2 | — | |
YQGUQZWOHCDPTK
|
7.3 | IC50 | 2 | — | |
JLUXEIBYLLFPTR
|
7.3 | IC50 | 2 | — | |
TVOBCJAKLFDOFL
|
7.3 | IC50 | 3 | — | |
YHVHYWYQEFELOW
|
7.3 | IC50 | 44 | — | |
ZOEILZXFYPPMTR
|
7.3 | IC50 | 2 | — | |
NGJAXUZGEAUCFH
|
7.3 | IC50 | 4 | — | |
ADCDBRPCQQHZQR
|
7.3 | IC50 | 2 | — | |
AEQQTRGTUZUWBY
|
7.3 | IC50 | 2 | — | |
AGGJFPXHGOZHPV
|
7.3 | IC50 | 2 | — | |
AHWSJOBFFQBHOW
|
7.3 | IC50 | 2 | — | |
ALNVGNKIGFPGCV
|
7.3 | IC50 | 3 | — | |
ANINHDBXZARAPZ
|
7.3 | IC50 | 2 | — |