Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NYVKAJAAGDOYJD
|
7.5 | IC50 | 3 | — | |
RSCAIJXVGDMQRL
|
7.5 | IC50 | 4 | — | |
BSBDXSGQMHVOLT
|
7.5 | IC50 | 2 | — | |
GCDSDVNITVBCDW
|
7.5 | IC50 | 17 | — | |
GLMRPQOSTRSLOB
|
7.5 | IC50 | 4 | — | |
GRUNJVATCGAOIE
|
7.5 | IC50 | 2 | — | |
LQGKYOJJBCEELL
|
7.5 | IC50 | 3 | — | |
RYQKZEFCGLDZCP
|
7.5 | IC50 | 2 | — | |
CBYOWSXIVYUEKV
|
7.5 | IC50 | 4 | — | |
FKZLDSCDUWVAGZ
|
7.5 | IC50 | 3 | — | |
HXIJRRHSUDWRPM
|
7.5 | IC50 | 2 | — | |
HZRWXAYRYYKKBH
|
7.5 | IC50 | 2 | — | |
QUNDXUVTKODMCV
|
7.5 | IC50 | 2 | — | |
QYRKJPSVGUQMLW
|
7.5 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
7.5 | Kd | 289 | Yes | |
UYSWRVPXWRGZTG
|
7.5 | IC50 | 4 | — | |
WORRXRIVSMTSEB
|
7.5 | IC50 | 4 | — | |
DOZGBVACZUIYTC
|
7.5 | IC50 | 3 | — | |
SZWMZMVQRXLMGH
|
7.5 | IC50 | 2 | — | |
TXIMZOFTQNLATM
|
7.5 | IC50 | 3 | — | |
ZTFAJUAGQGVBCO
|
7.5 | IC50 | 3 | — | |
FQNMCPIFXMICFV
|
7.5 | IC50 | 2 | — | |
HWAJPBLFIVLBGO
|
7.5 | IC50 | 3 | — | |
RXNGZWXHXININL
|
7.5 | IC50 | 3 | — | |
UFCSFQQMMHEHHY
|
7.5 | IC50 | 2 | — | |
ARSCEEUSPNVXQA
|
7.5 | IC50 | 4 | — | |
DYMOVSCTFZROSX
|
7.5 | IC50 | 3 | — | |
FQQXADKVHBKQJQ
|
7.5 | IC50 | 4 | — | |
GINRVSOEUKVVID
|
7.5 | IC50 | 2 | — | |
GPQKRDLDDKHLKK
|
7.5 | IC50 | 2 | — | |
IIDPZUKHHUHKFU
|
7.5 | IC50 | 3 | — | |
KQTRQDMQBAIPKT
|
7.5 | IC50 | 3 | — | |
NQFQOWLMRBYVBZ
|
7.5 | IC50 | 2 | — | |
QVWXQHOQYSJAID
|
7.5 | IC50 | 3 | — | |
FTNSEBXNCGRIEU
|
7.5 | IC50 | 4 | — | |
GBBCLTDGXQECOO
|
7.5 | IC50 | 4 | — | |
NCYONVSVKQVALR
|
7.5 | IC50 | 2 | — | |
PQKURPMJYNKLBD
|
7.5 | IC50 | 4 | — | |
APAJJMXZKHLSSS
|
7.4 | IC50 | 2 | — | |
LPVZJEBCLVVMCF
|
7.4 | IC50 | 2 | — | |
QXIOZIFTPMAING
|
7.4 | IC50 | 17 | — | |
RROWXJNEWORONQ
|
7.4 | IC50 | 3 | — | |
SOWKGLDGYDLSBM
|
7.4 | IC50 | 4 | — | |
WCBFHMOPYCFZQV
|
7.4 | IC50 | 2 | — | |
DVJHTWUZFJCMII
|
7.4 | IC50 | 2 | — | |
GEAJYTNNHUHUPD
|
7.4 | IC50 | 2 | — | |
MLIBDOUWSPIBHH
|
7.4 | IC50 | 4 | — | |
QEWWRQLOXCSNGA
|
7.4 | IC50 | 2 | — | |
QPIHEOATRHIZAP
|
7.4 | IC50 | 2 | — | |
STGJRXCRLCYESQ
|
7.4 | IC50 | 3 | — |