Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JYSXNODIVIMDDT
|
8.0 | IC50 | 2 | — | |
KRMIHQSNGSJHDA
|
8.0 | IC50 | 2 | — | |
LOONVQWRKJLEEG
|
8.0 | IC50 | 8 | — | |
MJKYJDTWPAMHCX
|
8.0 | IC50 | 4 | — | |
MTRDTDABXBDOPS
|
8.0 | IC50 | 4 | — | |
PFBFUNWWEQQNQB
|
8.0 | IC50 | 4 | — | |
SCCZGJNJWOJDLN
|
8.0 | IC50 | 4 | — | |
URJHRMXSWREGLT
|
8.0 | IC50 | 2 | — | |
XTKBOFNZDPSRBW
|
8.0 | IC50 | 2 | — | |
APMWOAUECKVBTF
|
7.9 | IC50 | 3 | — | |
DRBYDXGARLXEMD
|
7.9 | IC50 | 2 | — | |
DSZLKOXKYRREEO
|
7.9 | IC50 | 10 | — | |
HNYUGEZETOTTPJ
|
7.9 | IC50 | 3 | — | |
KVUCOURZIKDXHZ
|
7.9 | IC50 | 4 | — | |
PMMOUWGDKICRJR
|
7.9 | IC50 | 4 | — | |
QBCMBQCPRNSFJE
|
7.9 | IC50 | 3 | — | |
UGAWJRIPKFUXGB
|
7.9 | IC50 | 2 | — | |
YRANDDHDKOLWES
|
7.9 | IC50 | 2 | — | |
FLMRVDLSUJPCPS
|
7.9 | IC50 | 3 | — | |
HVRASXRMCOQSPI
|
7.9 | IC50 | 3 | — | |
OSSQCGAASUFADY
|
7.9 | IC50 | 2 | — | |
BIOCOIJRRXEMAB
|
7.9 | IC50 | 2 | — | |
CVMMQZHPZPFORW
|
7.9 | IC50 | 3 | — | |
NKPMZIRBMWWISL
|
7.9 | IC50 | 2 | — | |
OUOIQYPGNJQHIR
|
7.9 | IC50 | 4 | — | |
OWENAMOFXYZEJA
|
7.9 | IC50 | 4 | — | |
PTQDZIAZJFMTIT
|
7.9 | IC50 | 2 | — | |
QYWSJHPAXWONSF
|
7.9 | IC50 | 2 | — | |
XBFYWJOKBDZTSR
|
7.9 | IC50 | 4 | — | |
XMKLRDAMHIXNLW
|
7.9 | IC50 | 2 | — | |
DCZLCCHBIGHKPW
|
7.8 | IC50 | 3 | — | |
DERKWJPZXYTPTQ
|
7.8 | IC50 | 3 | — | |
JJIJUWUIPAWQRG
|
7.8 | IC50 | 4 | — | |
MXSXJVUUCUTMAN
|
7.8 | IC50 | 3 | — | |
QORFKFBKAXIHDO
|
7.8 | IC50 | 2 | — | |
RPDCDFMSBUBFCX
|
7.8 | IC50 | 4 | — | |
VNBRGSXVFBYQNN
|
7.8 | IC50 | 22 | Yes | |
XRLWMHNBPLXCKL
|
7.8 | IC50 | 2 | — | |
ZHHWIWQMTHPAOR
|
7.8 | IC50 | 2 | — | |
OBTYAQOWQNEKBT
|
7.8 | IC50 | 2 | — | |
UXHQCLFISGGSLE
|
7.8 | IC50 | 2 | — | |
VDZKYCXBCMIQDA
|
7.8 | IC50 | 5 | — | |
CLIUGIMDTBGMNI
|
7.8 | IC50 | 3 | — | |
CMXOTBPJJMRQOJ
|
7.8 | IC50 | 4 | — | |
CUDRWVZLQYDBKU
|
7.8 | IC50 | 4 | — | |
JRFAYFIOQCIYFZ
|
7.8 | IC50 | 2 | — | |
NEAJWUKNRWPSCI
|
7.8 | IC50 | 2 | — | |
POLOQBZTXAWWJT
|
7.8 | IC50 | 3 | — | |
SFMTZXDPBZEXMO
|
7.8 | IC50 | 2 | — | |
VFONQNZZLGMGFZ
|
7.8 | IC50 | 3 | — |