Target Details
| UniProt AC | Q12866 |
|---|---|
| Gene Symbol | MERTK |
| Protein Name | Tyrosine-protein kinase Mer |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00041 (fn3) PF00047 (ig) PF13927 (Ig_3) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 1,592
- Clinical molecules 13
- Avg pChEMBL 7.42
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (1,592)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VPEBETSCTWIJQZ
|
9.9 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
9.6 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
9.6 | Kd | 149 | — | |
FAOUZNFWHWLTIC
|
9.5 | IC50 | 3 | — | |
XWAYWHRXNQJWEN
|
9.4 | IC50 | 3 | — | |
IBLUITUCVORWLC
|
9.4 | IC50 | 3 | — | |
GMAFXYZWTSGYMU
|
9.4 | IC50 | 4 | — | |
KSZDMKRJEQNXAQ
|
9.4 | IC50 | 3 | — | |
IADRGGYOCXDICI
|
9.3 | IC50 | 4 | — | |
XGIIMGRAMUXNFL
|
9.3 | IC50 | 4 | — | |
UHQXCBSLWHQJJT
|
9.3 | IC50 | 2 | — | |
JNOZPOGAIWIGDX
|
9.3 | IC50 | 3 | — | |
HSJCSHDUINVROZ
|
9.2 | IC50 | 4 | — | |
DCFNMFYAKVXCLN
|
9.2 | IC50 | 4 | — | |
HOUOLCBDDCEYMO
|
9.2 | IC50 | 2 | — | |
HYUGTGGDEAGXJP
|
9.2 | IC50 | 11 | — | |
ZPXYYHKOOQSKHV
|
9.2 | IC50 | 4 | — | |
SINLAAVSJWFXNK
|
9.2 | IC50 | 4 | — | |
YHELBFBDLFOCAS
|
9.2 | IC50 | 4 | — | |
WERQRDFKILOXSK
|
9.2 | IC50 | 3 | — | |
WERQRDFKILOXSK
|
9.2 | IC50 | 4 | — | |
WZSUDZDKYJWJPS
|
9.2 | IC50 | 4 | — | |
WZSUDZDKYJWJPS
|
9.2 | IC50 | 3 | — | |
XEHHSTXCXVSYIR
|
9.2 | IC50 | 3 | — | |
ISOYAPPKZDNVQA
|
9.1 | IC50 | 3 | — | |
LWZKYWNWDTZZGI
|
9.1 | IC50 | 3 | — | |
ZYBHGENFQHMBLJ
|
9.1 | IC50 | 4 | — | |
GDKUSUOIODZPAK
|
9.1 | IC50 | 3 | — | |
DKZQQJXYLNUWFT
|
9.1 | IC50 | 4 | — | |
QHADVLVFMKEIIP
|
9.1 | IC50 | 9 | — | |
QIRBYYSKWYYQEJ
|
9.1 | IC50 | 3 | — | |
MDPKWYPYSBXZHN
|
9.1 | IC50 | 2 | — | |
NLXWFBBYANWXPR
|
9.1 | IC50 | 3 | — | |
NLXWFBBYANWXPR
|
9.1 | IC50 | 4 | — | |
RTZPWZZLLAHMAA
|
9.1 | IC50 | 4 | — | |
MSWOWUREQODTRO
|
9.1 | IC50 | 11 | — | |
WOVFEULIRSIJJU
|
9.1 | IC50 | 4 | — | |
XYSYRHAUHUPOHK
|
9.1 | IC50 | 4 | — | |
FGYMKXFFIWSCGZ
|
9.1 | IC50 | 4 | — | |
JTWJBADLHDCZDM
|
9.1 | IC50 | 3 | — | |
QEVGJXHJXPXEJA
|
9.1 | IC50 | 4 | — | |
RCQLJPMEVONOSW
|
9.1 | IC50 | 4 | — | |
FEXRSRXFBIRFMY
|
9.0 | IC50 | 4 | — | |
YLCUJYLNOPDSFV
|
9.0 | IC50 | 3 | — | |
BWLVWHQFWOPSOP
|
9.0 | IC50 | 4 | — | |
MIYIUVBGBPRNLG
|
9.0 | IC50 | 4 | — | |
LBEJYFVJIPQSNX
|
9.0 | IC50 | 4 | — | |
SLCVMWQKWVHPQE
|
9.0 | IC50 | 3 | — | |
FECNHZJRCCTFMT
|
9.0 | IC50 | 2 | — | |
HDRSWNSYJOUCLI
|
9.0 | IC50 | 3 | — |