Target Details
| UniProt AC | Q12852 |
|---|---|
| Gene Symbol | MAP3K12 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 12 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 54
- Clinical molecules 8
- Avg pChEMBL 7.47
KEGG Pathways (1)
Active Molecules (54)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZNLWKSRHKZKBQH
|
9.9 | Kd | 2 | — | |
LYWYGIOUJQXFNS
|
9.8 | Ki | 2 | — | |
MZUKCHWHYOQJRJ
|
9.4 | Ki | 2 | — | |
JKALQBFVHDTVCS
|
8.7 | IC50 | 2 | — | |
OYNJYGXCFZHONL
|
8.7 | IC50 | 2 | — | |
APYQWPISTZCVOT
|
8.5 | IC50 | 2 | — | |
KBBJVNCJPHHXME
|
8.5 | IC50 | 2 | — | |
WQQYNNJZQBRUAR
|
8.5 | IC50 | 2 | — | |
SKMKJBYBPYBDMN
|
8.5 | IC50 | 3 | — | |
CMXUWUGBGXEFFR
|
8.4 | IC50 | 3 | — | |
LDWXXJNYXNYPRY
|
8.4 | IC50 | 2 | — | |
PDNZDVAQMFNPMG
|
8.4 | IC50 | 2 | — | |
IRPVABHDSJVBNZ
|
8.3 | Ki | 6 | — | |
UHEFRVBGJORHNV
|
8.0 | IC50 | 4 | — | |
IQLAMFMVULXILA
|
7.9 | IC50 | 2 | — | |
AKKHHVJIISFQCL
|
7.9 | IC50 | 2 | — | |
BURDQUKVCPYGRG
|
7.9 | Kd | 3 | — | |
CQPIBQJUQSJKOA
|
7.9 | IC50 | 2 | — | |
XYWGNKCGTAROOP
|
7.9 | IC50 | 2 | — | |
GYENDIAEYZIMIV
|
7.8 | IC50 | 2 | — | |
AVWDJSXSWJBVBP
|
7.8 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
7.7 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.7 | Kd | 149 | — | |
FSNRHEHUJCWRAQ
|
7.6 | IC50 | 2 | — | |
HCDVOAGDQONFDT
|
7.6 | Ki | 4 | — | |
GIRIQGHXPJDILQ
|
7.5 | IC50 | 2 | — | |
RHFIAUKMKYHHFA
|
7.5 | IC50 | 9 | — | |
QQWUGDVOUVUTOY
|
7.4 | Kd | 231 | Yes | |
PWQYILBUZALMLM
|
7.3 | IC50 | 2 | — | |
AVWDJSXSWJBVBP
|
7.3 | IC50 | 2 | — | |
QUJWSXIGZUDUAB
|
7.3 | IC50 | 2 | — | |
AKKHHVJIISFQCL
|
7.2 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
UOWUCCPLVGOHMV
|
7.1 | IC50 | 2 | — | |
JAXBPMVTQNGQOE
|
7.0 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
7.0 | Kd | 201 | Yes | |
GEXWJSDYWQNHLQ
|
7.0 | Ki | 2 | — | |
XZXHXSATPCNXJR
|
6.8 | Kd | 165 | Yes | |
VBUUATKGJOATLP
|
6.8 | Ki | 2 | — | |
KTEIFNKAUNYNJU
|
6.8 | Kd | 114 | — | |
HKSZLNNOFSGOKW
|
6.8 | IC50 | 408 | — | |
GCIKSSRWRFVXBI
|
6.7 | Kd | 109 | Yes | |
XGFVOKJJQCQLJX
|
6.7 | IC50 | 2 | — | |
HTNKTPXNQZIMGF
|
6.6 | Ki | 2 | — | |
GUBJNPWVIUFSTR
|
6.5 | Kd | 103 | — | |
JWNPDZNEKVCWMY
|
6.4 | Kd | 57 | Yes | |
CTNPALGJUAXMMC
|
6.2 | Kd | 151 | — | |
OYONTEXKYJZFHA
|
6.2 | Kd | 69 | Yes | |
UBPYILGKFZZVDX
|
6.2 | Kd | 130 | Yes | |
WUQFEMGACGWUFQ
|
6.2 | Ki | 2 | — |