Target Details
| UniProt AC | Q12851 |
|---|---|
| Gene Symbol | MAP4K2 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 326
- Clinical molecules 25
- Avg pChEMBL 6.89
KEGG Pathways (1)
Active Molecules (326)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PPCNMZPSQZFFGM
|
6.1 | Ki | 8 | — | |
RUPJOKGREQMQSI
|
6.1 | Ki | 9 | — | |
UMYBAQLXZPEUQW
|
6.1 | Ki | 15 | — | |
URNZTLZSAVLTIZ
|
6.1 | Ki | 26 | — | |
VLEFVPMCVJDTHZ
|
6.1 | Ki | 13 | — | |
VVEGARMQKNYDID
|
6.1 | Ki | 24 | — | |
XMGFTZYNTYNOOJ
|
6.1 | Ki | 10 | — | |
YYPKOMNJRZRWIC
|
6.1 | Ki | 26 | — | |
BLLJUCXNHUVEHL
|
6.1 | IC50 | 3 | — | |
AFUHWZUYZJGVKM
|
6.0 | Kd | 5 | — | |
FCMKRDBRBZALAL
|
6.0 | IC50 | 2 | — | |
AAYZTFLAQXDFOL
|
6.0 | Ki | 11 | — | |
BIIVYFLTOXDAOV
|
6.0 | Ki | 31 | — | |
FAIHBCXQSBIRIL
|
6.0 | Ki | 22 | — | |
GNLAGGCSJGJECE
|
6.0 | Ki | 19 | Yes | |
GQLWKGVBOIYMTN
|
6.0 | Ki | 35 | — | |
HRZOUBQYVUXBNS
|
6.0 | Ki | 38 | — | |
HSMUWLLZAZCLHF
|
6.0 | Ki | 25 | — | |
IBPSHHSPUPWXHN
|
6.0 | Ki | 6 | — | |
JBRASADWXDKCLJ
|
6.0 | Ki | 22 | — | |
NECQZMQPXFYVOY
|
6.0 | Ki | 26 | — | |
SEVCBWKJSOLMNQ
|
6.0 | Ki | 38 | — | |
WAKGEHXTOOFEAE
|
6.0 | Ki | 27 | — | |
XFCOCCMXXFTEEC
|
6.0 | Ki | 6 | — | |
XJJYJNMNYDNXNO
|
6.0 | Ki | 23 | — | |
ZYTFPHRVOZXPGZ
|
6.0 | Ki | 30 | — |