Target Details
| UniProt AC | Q12851 |
|---|---|
| Gene Symbol | MAP4K2 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 326
- Clinical molecules 25
- Avg pChEMBL 6.89
KEGG Pathways (1)
Active Molecules (326)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IJNGXROUMFEKDB
|
6.3 | Ki | 39 | — | |
ILUGAYBMBIJXHC
|
6.3 | Ki | 9 | — | |
ISVHLTLEHRZKJC
|
6.3 | Ki | 19 | — | |
JHYHWHUTTXJICB
|
6.3 | Ki | 18 | — | |
KNRKFYBCACDGCC
|
6.3 | IC50 | 2 | — | |
MADCXGNPDBWPLM
|
6.3 | Ki | 25 | — | |
NKEUPUJTVALZIK
|
6.3 | Ki | 28 | — | |
NWAUBAGBGOPJLF
|
6.3 | Ki | 51 | Yes | |
NXNQLECPAXXYTR
|
6.3 | Ki | 29 | — | |
OWDRQHVEJIYVOI
|
6.3 | Ki | 47 | — | |
QVNZKVACBBTKSL
|
6.3 | Ki | 38 | — | |
RIUZPIBUSOHUKF
|
6.3 | Ki | 23 | — | |
RWEHAHIEUDLKGT
|
6.3 | Ki | 33 | — | |
SFPWNTQWFFNJIH
|
6.3 | Ki | 48 | — | |
UGUZOLHBLLTLBA
|
6.3 | Ki | 15 | — | |
XNEPVLVYFUGJLF
|
6.3 | Ki | 27 | — | |
XXSPHNFKLDJDAK
|
6.3 | Ki | 26 | — | |
XYXLUJQBBIBJFV
|
6.3 | Ki | 36 | — | |
YKJSWMAVAKRUAN
|
6.3 | Ki | 19 | — | |
HUAPVUVLSXALII
|
6.3 | IC50 | 3 | — | |
XXJWYDDUDKYVKI
|
6.3 | Kd | 52 | — | |
SUBYPZBREZXPCW
|
6.2 | IC50 | 3 | — | |
VNADJTWHOAMTLY
|
6.2 | Kd | 4 | — | |
WOSKHXYHFSIKNG
|
6.2 | Kd | 24 | — | |
XCOSAQGGGZDYJN
|
6.2 | IC50 | 11 | — | |
ATGVCJYHNOSZEV
|
6.2 | Ki | 23 | — | |
CHADTINFLWZSKR
|
6.2 | Ki | 26 | — | |
DLWMVUDMPMKGEE
|
6.2 | Ki | 24 | — | |
GJKVMXDBPDDFHI
|
6.2 | Ki | 27 | — | |
LJKJYKWDLJUZHA
|
6.2 | Ki | 24 | — | |
MIYRKQLKDQNUKZ
|
6.2 | Ki | 23 | — | |
OQSVYNYDHYYKJX
|
6.2 | Ki | 7 | — | |
PBCZSGKMGDDXIJ
|
6.2 | Kd | 68 | Yes | |
PIQCTGMSNWUMAF
|
6.2 | Ki | 137 | Yes | |
PUPCRRRSBUYJAD
|
6.2 | Ki | 44 | Yes | |
SKKRZILJUKYLJS
|
6.2 | Ki | 25 | — | |
TZSJMSZEKQGCBI
|
6.2 | Ki | 15 | — | |
UNVKXVCDLOLPJE
|
6.2 | Ki | 8 | — | |
UWDBNTXEKYRMSG
|
6.2 | Ki | 26 | — | |
XSDJOIOVIMPMHD
|
6.2 | Ki | 44 | — | |
NHHQJBCNYHBUSI
|
6.2 | Kd | 220 | — | |
HXHAJRMTJXHJJZ
|
6.1 | Kd | 52 | Yes | |
AOBLBPWPSKBHSI
|
6.1 | Ki | 55 | — | |
AQQWWOMMPDCTLW
|
6.1 | Ki | 10 | — | |
BRTHUECZMVKNMQ
|
6.1 | Ki | 31 | — | |
FPQHXFMYXQZPSV
|
6.1 | Ki | 23 | — | |
HHSVICUMCOBRPT
|
6.1 | Ki | 33 | — | |
JJJSCYSPSKBQAX
|
6.1 | Ki | 34 | — | |
MZIOLOXGGOLJMJ
|
6.1 | Ki | 12 | — | |
PKCDDUHJAFVJJB
|
6.1 | Ki | 13 | — |