Target Details
UniProt ACQ12851
Gene SymbolMAP4K2
Protein NameMitogen-activated protein kinase kinase kinase kinase 2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00780 (CNH) PF00069 (Pkinase)
Summary
  • Multi-target molecules 326
  • Clinical molecules 25
  • Avg pChEMBL 6.89
KEGG Pathways (1)
Top Co-occurrence Targets
Active Molecules (326)
InChIKey pChEMBL Type Targets Clinical
NVRXTLZYXZNATH 6.5 Ki 47 Yes
RITAVMQDGBJQJZ 6.5 Ki 33
RTYJMUXLFRYRBU 6.5 Ki 35
SBFPHSVZEXSHTL 6.5 Ki 62
TVLFEDKEAOXRCZ 6.5 Ki 22
UYGYYOIUVFMGKQ 6.5 Ki 30
VSVWQTDDGQSGHP 6.5 Ki 51
VXYDJXMHISGSDA 6.5 Ki 59
WZISGNDZZPSYRP 6.5 Ki 20
XAHJIRNRDAKTEF 6.5 Ki 18
XNWKXXIGSPPPBH 6.5 Ki 31
XUFLBSMTYMFOQH 6.5 Ki 43
YUOWJICKAJQZLS 6.5 Ki 35
ZKHDDJKHTPLPOQ 6.5 Ki 62
ZWVZORIKUNOTCS 6.5 Ki 69
OMZCMEYTWSXEPZ 6.5 Kd 43 Yes
LGIBDQRYOFBMTC 6.5 Ki 6 Yes
ALKJNCZNEOTEMP 6.5 Kd 55
YXFNNHJWPFANTQ 6.5 IC50 3
APPXQUDJLJXULP 6.4 IC50 47
ACSYKUPGCXYRRO 6.4 Ki 26
AEYLJTAIDDIOBA 6.4 Ki 53
HAYYBYPASCDWEQ 6.4 Ki 47
IFPPYSWJNWHOLQ 6.4 Ki 52 Yes
KYACBMRLQMEIAI 6.4 Ki 30
LXVBELDBJGYFEM 6.4 Ki 20
MASJMHFQMYAPJR 6.4 Ki 41
MFMXAWQGPQXDRJ 6.4 Ki 27
MHWHPWMWKYXCRJ 6.4 Ki 32
NRGYZNJPCGRCLV 6.4 Ki 52
OEEGUWWPGAZRIJ 6.4 Ki 21
PNKALLUVKOKYHZ 6.4 Ki 32
QAJPIJHWTGPUNZ 6.4 Ki 37
QBKUOOQFSVMDPB 6.4 Ki 31
QNUKRWAIZMBVCU 6.4 Ki 46
SRONQUHCRFZABC 6.4 Ki 28
UOVCGJXDGOGOCZ 6.4 Ki 59
UQNNJYLAPYGZBD 6.4 Ki 28
XKFTZKGMDDZMJI 6.4 Ki 56
ZDPGLLQANLROFM 6.4 Ki 17
ZGZVRPRSFXRGCF 6.4 Ki 76
ZVWRFVCNQOECJS 6.4 Ki 71
ZXLFIHLBHMLHFJ 6.4 Ki 31
HENRITOGWFFGGA 6.3 IC50 2
ACNCCUVYXQGPKZ 6.3 Ki 31
DKSNLQYRZJKYOC 6.3 Ki 51
GHMRUNOHAHJNNA 6.3 Ki 29
GJOXRIYWDHESDF 6.3 Ki 27
HKZKELVPGXJIMW 6.3 Ki 41
HZPACYSNLOCDLW 6.3 Ki 48
2D structure