Target Details
| UniProt AC | Q12851 |
|---|---|
| Gene Symbol | MAP4K2 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 326
- Clinical molecules 25
- Avg pChEMBL 6.89
KEGG Pathways (1)
Active Molecules (326)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XHORJSJFHVABEA
|
6.9 | Ki | 49 | — | |
ZLVOTRRGLSDLPF
|
6.9 | Ki | 36 | — | |
KOZFSFOOLUUIGY
|
6.9 | Kd | 88 | Yes | |
AUDNGNGLLRZLDR
|
6.8 | Ki | 33 | — | |
CQBBMNXXVMOFCA
|
6.8 | Ki | 39 | — | |
MHCPAORAYMTGCZ
|
6.8 | Ki | 37 | — | |
OWFXKTOLFUQPDJ
|
6.8 | Ki | 36 | — | |
PSCJSWRVCKUMSL
|
6.8 | Ki | 35 | — | |
PUYIXDDMOUMMRR
|
6.8 | Ki | 27 | — | |
DKZYXHCYPUVGAF
|
6.8 | Kd | 112 | — | |
FJABJYQHNWUFPP
|
6.8 | IC50 | 2 | — | |
OFGWSAWNQPAURN
|
6.8 | IC50 | 2 | — | |
IVUGFMLRJOCGAS
|
6.7 | Kd | 9 | — | |
QQWUGDVOUVUTOY
|
6.7 | Kd | 231 | Yes | |
DCTBPIBEQFLAOQ
|
6.7 | Ki | 13 | — | |
KOHNRDPXFDZZJF
|
6.7 | Ki | 31 | — | |
KTWBYGUSEYSRND
|
6.7 | Ki | 28 | — | |
LCHCSKHPVCDXAU
|
6.7 | Ki | 30 | — | |
PLHUMPJXRHMFFR
|
6.7 | Ki | 28 | — | |
QONPPIZSNSSCSK
|
6.7 | Ki | 45 | Yes | |
RKUKAACYUCUJEE
|
6.7 | Ki | 58 | — | |
UUWNXFJBBYAMDT
|
6.7 | Ki | 46 | — | |
JWNPDZNEKVCWMY
|
6.7 | Kd | 57 | Yes | |
WVXNSAVVKYZVOE
|
6.6 | IC50 | 92 | — | |
XCAXLCSQKKQKHA
|
6.6 | IC50 | 3 | — | |
DFMCXVONDDGQIY
|
6.6 | Ki | 66 | — | |
NFMGZVPRGVERNN
|
6.6 | Ki | 44 | — | |
PROLIXHVRCJEFH
|
6.6 | Ki | 46 | — | |
PTVPBWWDGZSEAF
|
6.6 | Ki | 63 | — | |
RFBPWKMQWSIPEO
|
6.6 | Ki | 28 | — | |
RYAVJHIPOWNWDE
|
6.6 | Ki | 38 | — | |
UIRCQOKSJDLYBB
|
6.6 | Ki | 50 | — | |
VTQQYBGURNVVFE
|
6.6 | Ki | 17 | — | |
WQFGNANQTYLQBP
|
6.6 | Ki | 16 | — | |
ZGDYBJXDIXVTLV
|
6.6 | Ki | 54 | — | |
XKFTZKGMDDZMJI
|
6.6 | Kd | 64 | Yes | |
KTEIFNKAUNYNJU
|
6.5 | Ki | 48 | — | |
XZXHXSATPCNXJR
|
6.5 | Kd | 165 | Yes | |
ZCBUQCWBWNUWSU
|
6.5 | Kd | 59 | — | |
OLKMNKWCYPTDSI
|
6.5 | IC50 | 2 | — | |
AQZIXHSRFOGYHF
|
6.5 | Ki | 9 | — | |
CNTCGRJDUJEUDG
|
6.5 | Ki | 37 | — | |
FXQWJULRETZHHW
|
6.5 | Ki | 14 | — | |
GCZJQTRRJPRFIP
|
6.5 | Ki | 10 | — | |
GSXRCPJTNIGKSZ
|
6.5 | Ki | 43 | — | |
KIUHBHFVVQQALF
|
6.5 | Ki | 9 | — | |
KUNZDWIFPOMUOX
|
6.5 | Ki | 36 | — | |
LGHBDVLAHHANMX
|
6.5 | Ki | 53 | — | |
MTCHQDWUHQADSY
|
6.5 | Ki | 29 | — | |
NOBMKUVHFRVBES
|
6.5 | Ki | 19 | — |