Target Details
| UniProt AC | Q12851 |
|---|---|
| Gene Symbol | MAP4K2 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 326
- Clinical molecules 25
- Avg pChEMBL 6.89
KEGG Pathways (1)
Active Molecules (326)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NJPWCTYVEJIQBM
|
7.2 | Ki | 72 | — | |
QPORZABOFXPRHM
|
7.2 | Ki | 18 | — | |
TVUWQDLBEOZVOU
|
7.2 | Ki | 41 | — | |
UEEVERDPEVIFBH
|
7.2 | IC50 | 2 | — | |
UMTWTCVTRDYHQQ
|
7.2 | Ki | 56 | — | |
WDARYLSSWBWVCU
|
7.2 | Ki | 49 | — | |
XBYVOPRDASFDMY
|
7.2 | Ki | 42 | — | |
XCHWBXBDZRJVDP
|
7.2 | Ki | 51 | — | |
GUBJNPWVIUFSTR
|
7.2 | Kd | 103 | — | |
PKCDDUHJAFVJJB
|
7.2 | Kd | 13 | — | |
PIMBZWQACDWQJV
|
7.1 | IC50 | 2 | — | |
AIQDZMUPVYDVLB
|
7.1 | Ki | 48 | — | |
CFIBXVQLBVNOHW
|
7.1 | Ki | 64 | — | |
CNQGNADBGYCKKV
|
7.1 | Ki | 25 | — | |
DTMZXHDQZQLTHA
|
7.1 | Ki | 21 | — | |
GDYZFFBMSBDTAA
|
7.1 | Ki | 60 | — | |
KNACLJBHKVSTDL
|
7.1 | Ki | 40 | — | |
KTEIFNKAUNYNJU
|
7.1 | Kd | 114 | — | |
LRLDYTTWQIFWBD
|
7.1 | Ki | 25 | — | |
NZVDDFRUBIEKLV
|
7.1 | Ki | 20 | — | |
RGNHKJWHFIPHIM
|
7.1 | Ki | 66 | — | |
SMRWVXLSRJWVBF
|
7.1 | Ki | 25 | — | |
UDFDIIVNIYWXDM
|
7.1 | Ki | 74 | — | |
VWACUNWBMWWMPJ
|
7.1 | Ki | 18 | — | |
XKZQZMSAWVDRSP
|
7.1 | Ki | 39 | Yes | |
XPHWIERLJBFPFV
|
7.1 | Ki | 69 | — | |
BIIVYFLTOXDAOV
|
7.0 | Kd | 82 | Yes | |
UMBFDGUGXMOMHX
|
7.0 | IC50 | 12 | — | |
BIKYDWLMTPRSQL
|
7.0 | Ki | 50 | — | |
LVECPYVAIBNSRV
|
7.0 | Ki | 33 | — | |
MFAQYJIYDMLAIM
|
7.0 | Kd | 130 | Yes | |
ODPGGGTTYSGTGO
|
7.0 | Kd | 153 | — | |
OLVBAUVSICCWEJ
|
7.0 | Ki | 39 | — | |
ULHGAQSVFPOUDY
|
7.0 | Ki | 43 | — | |
VKBFHTIUXUCYRQ
|
7.0 | Ki | 66 | — | |
VUHZDNOPEVGHEO
|
7.0 | Ki | 29 | — | |
XSRHBCYNCKAFKS
|
7.0 | Ki | 45 | — | |
JKHBVOCOHYSWTQ
|
7.0 | IC50 | 3 | — | |
VRQMAABPASPXMW
|
7.0 | Kd | 10 | — | |
UJBJWYNPUOLFIZ
|
6.9 | IC50 | 49 | — | |
DSSNAGYVGTYAGH
|
6.9 | IC50 | 10 | — | |
ONPGOSVDVDPBCY
|
6.9 | Kd | 2 | — | |
ADLPKFFMGIJZIM
|
6.9 | Ki | 44 | — | |
CZQVOIDVDAVDFW
|
6.9 | Ki | 18 | — | |
DBXGGXLBTWZXBB
|
6.9 | Ki | 39 | — | |
DPEXRCOBPACFOO
|
6.9 | Ki | 36 | — | |
LRINYHMQZRENCY
|
6.9 | Ki | 29 | — | |
MQRDVGBWWVWMEN
|
6.9 | Ki | 47 | — | |
OLUKILHGKRVDCT
|
6.9 | Ki | 44 | Yes | |
SLKCVFPEQGHNSI
|
6.9 | Ki | 29 | — |