Target Details
| UniProt AC | Q12851 |
|---|---|
| Gene Symbol | MAP4K2 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 326
- Clinical molecules 25
- Avg pChEMBL 6.89
KEGG Pathways (1)
Active Molecules (326)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GZYCQQBRSRIFII
|
7.6 | Kd | 7 | — | |
IZAVTOABECKIDH
|
7.6 | Ki | 20 | — | |
YDWMUCKJUNLURC
|
7.6 | Ki | 24 | — | |
YWTBGJGMTBHQTM
|
7.6 | Ki | 65 | — | |
JIOOBLLPEPCAAJ
|
7.6 | IC50 | 4 | — | |
HMVDGWSYIBOKRV
|
7.6 | IC50 | 2 | — | |
ZWVLMQTXUWMUII
|
7.5 | IC50 | 9 | Yes | |
AMHWQBGAKJESFB
|
7.5 | IC50 | 4 | — | |
FCNPQYHKUYSELK
|
7.5 | IC50 | 8 | — | |
DQPYZHUAILXFJI
|
7.5 | Ki | 27 | — | |
MCCCQFAOMZMZKE
|
7.5 | Ki | 52 | — | |
SDBOIBYRBWPIEL
|
7.5 | Ki | 31 | — | |
XOOAAYRIVATZNM
|
7.5 | Ki | 55 | — | |
AQVOAZGKJLFRRO
|
7.5 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
7.5 | Kd | 201 | Yes | |
PESNFBOGJFKUMG
|
7.5 | IC50 | 2 | — | |
PWPDYURZGAQWPZ
|
7.4 | IC50 | 2 | — | |
BSFNGHCTZDCQBF
|
7.4 | Ki | 93 | — | |
FUMCKNCUEAQHCV
|
7.4 | Ki | 103 | — | |
HEUSUIRCBWROMH
|
7.4 | Ki | 64 | — | |
KWRXWPRFIUJQBP
|
7.4 | Ki | 25 | — | |
LACOMQAWPSFXQC
|
7.4 | Ki | 27 | — | |
MCKPYPWHBUXLEZ
|
7.4 | Ki | 21 | — | |
RWKDVIAVTRRJIR
|
7.4 | Ki | 23 | — | |
RYYNGWLOYLRZLK
|
7.4 | Ki | 104 | — | |
UAQJVFADAYIBGC
|
7.4 | Ki | 23 | — | |
VCZPJHYQIPIKSV
|
7.4 | IC50 | 3 | — | |
XJSFDMGICAWQFS
|
7.4 | Ki | 60 | — | |
PHXJVRSECIGDHY
|
7.4 | Kd | 59 | — | |
NEIVLVMGHRRCDM
|
7.4 | IC50 | 2 | — | |
XLFJEGWLJGWRSM
|
7.4 | IC50 | 4 | — | |
GGGQYLRXTXDJRN
|
7.3 | IC50 | 2 | — | |
JWXZQEPPXRGVKZ
|
7.3 | IC50 | 3 | — | |
PCFQERXLBAHWRY
|
7.3 | IC50 | 4 | — | |
ADMFLILDQJSEIK
|
7.3 | Ki | 72 | — | |
BGYVWFZMYBWCNY
|
7.3 | Ki | 30 | — | |
GUMBHNMWKMFKRT
|
7.3 | Ki | 23 | — | |
HOYRWTWZUFFACV
|
7.3 | Ki | 28 | — | |
IAYGCINLNONXHY
|
7.3 | Kd | 50 | — | |
JOGKUKXHTYWRGZ
|
7.3 | Ki | 28 | — | |
KRIUNPBAQZGFQA
|
7.3 | Ki | 76 | — | |
LPILBMJJRGTKOQ
|
7.3 | Ki | 27 | — | |
ZGGIYFOLDBTZIL
|
7.3 | Ki | 27 | — | |
DFHIKCGHCSDYRT
|
7.3 | IC50 | 2 | — | |
LAJAFFLJAJMYLK
|
7.2 | IC50 | 17 | — | |
BPNUQXPIQBZCMR
|
7.2 | Ki | 60 | — | |
CHTMRWQLNNRRFJ
|
7.2 | Ki | 70 | — | |
IAKGNUWZPSPEKU
|
7.2 | Ki | 19 | — | |
MULNSLQVKKUPJN
|
7.2 | Ki | 41 | — | |
MVJMMLFMPWITEJ
|
7.2 | Ki | 110 | — |