Target Details
| UniProt AC | Q12851 |
|---|---|
| Gene Symbol | MAP4K2 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 326
- Clinical molecules 25
- Avg pChEMBL 6.89
KEGG Pathways (1)
Active Molecules (326)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FCMNXGJPIJFWQV
|
9.0 | IC50 | 2 | — | |
BJKWAQGXAVDGLG
|
8.7 | IC50 | 2 | — | |
KHGPYYFCIAISBU
|
8.7 | Ki | 31 | — | |
REEJHXFEIZURCB
|
8.7 | IC50 | 2 | — | |
YMIJUBCSOKSFRU
|
8.5 | Ki | 87 | — | |
ZKLJKKASNXVQBZ
|
8.5 | Ki | 27 | — | |
UIARLYUEJFELEN
|
8.3 | Kd | 289 | Yes | |
FZPWJZCQBCBZKE
|
8.3 | IC50 | 2 | — | |
GCBJDOWIQHMCMR
|
8.3 | Ki | 84 | — | |
HKSZLNNOFSGOKW
|
8.3 | Ki | 118 | — | |
NBZFRTJWEIHFPF
|
8.3 | IC50 | 3 | — | |
RJZDECGDCKOHBV
|
8.3 | Ki | 70 | — | |
KNRXPUFRSHTQJW
|
8.2 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
8.2 | Kd | 200 | — | |
GWFZRGVIOWEPRA
|
8.2 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
8.2 | Kd | 170 | — | |
FLEAYYMORDPWAJ
|
8.1 | Ki | 90 | — | |
GCYXEGSPUDSZJY
|
8.1 | Ki | 82 | — | |
OUJZYQBEFNDJQN
|
8.1 | Ki | 71 | — | |
SZNYUUZOQHNEKB
|
8.1 | IC50 | 7 | — | |
VPOWOPVCLUEIIA
|
8.1 | IC50 | 2 | — | |
WPHKIQPVPYJNAX
|
8.1 | Ki | 81 | — | |
HKSZLNNOFSGOKW
|
8.1 | Kd | 408 | — | |
OHBDADSLOSGAHB
|
8.0 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
8.0 | Kd | 130 | Yes | |
WSTUJEXAPHIEIM
|
8.0 | Kd | 10 | — | |
YYLKKYCXAOBSRM
|
8.0 | Kd | 191 | — | |
ZCCPLJOKGAACRT
|
7.9 | Kd | 599 | — | |
RBXYGQNZRVPDNB
|
7.9 | Ki | 34 | — | |
MWKSRKSEWLRPBL
|
7.9 | Kd | 1075 | — | |
BIMOMBRKBARWLJ
|
7.8 | IC50 | 2 | — | |
IFRQDJZBFXKVOQ
|
7.8 | IC50 | 2 | — | |
JWQOJVOKBAAAAR
|
7.8 | Ki | 29 | — | |
LSLPDHNUWRDOGC
|
7.8 | Ki | 25 | — | |
NWMPVMMGSHXANZ
|
7.8 | Ki | 58 | — | |
YEHCNYAQEBQCCS
|
7.8 | Ki | 74 | — | |
USVYVEUGCBHMNU
|
7.8 | IC50 | 2 | — | |
RWNAOXLCVXJMGM
|
7.7 | IC50 | 5 | — | |
ASCPSRDSSMPJDW
|
7.7 | IC50 | 3 | — | |
JZTOUVBEZONDKA
|
7.7 | Ki | 80 | — | |
LYNBNVBMAGDJRW
|
7.7 | Ki | 81 | — | |
NLUPJKQOKWBWFC
|
7.7 | Ki | 69 | — | |
OADRBDVURCEKRP
|
7.7 | Ki | 44 | — | |
VCFDMLBPASGZTP
|
7.7 | Ki | 38 | — | |
XKZINYYXWJEYEL
|
7.7 | Ki | 37 | — | |
PPCIDOUXWYIBPO
|
7.7 | IC50 | 6 | — | |
SMPGEBOIKULBCT
|
7.7 | IC50 | 15 | — | |
GNIYUURCQFKRCB
|
7.6 | IC50 | 11 | Yes | |
OHPMDANXCFNAPB
|
7.6 | IC50 | 2 | — | |
RPDGGTQIKZCYAP
|
7.6 | IC50 | 3 | — |