Target Details
| UniProt AC | Q12830 |
|---|---|
| Gene Symbol | BPTF |
| Protein Name | Nucleosome-remodeling factor subunit BPTF |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00439 (Bromodomain) PF02791 (DDT) PF00628 (PHD) PF15613 (WSD) |
Summary
- Multi-target molecules 10
- Clinical molecules 0
- Avg pChEMBL 6.96
Active Molecules (10)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CIUXKWFQVPTMEQ
|
7.7 | IC50 | 3 | — | |
UOQAFGWMKNIVAR
|
7.7 | IC50 | 6 | — | |
RORQWFZBNDBULQ
|
7.2 | IC50 | 3 | — | |
JYTISQGEFSHUIR
|
7.2 | Kd | 4 | — | |
RBUYFHLQNPJMQM
|
7.0 | Kd | 10 | — | |
VZAFGXCWAWRULT
|
6.9 | Ki | 7 | — | |
MSIJJXOWLFOYIN
|
6.7 | Kd | 2 | — | |
OHVGMQWGTYKZJL
|
6.7 | IC50 | 2 | — | |
GXHSEYWYHGZDGJ
|
6.6 | IC50 | 2 | — | |
PUFPGLSWMMJNSE
|
6.0 | Kd | 3 | — |