Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KPJNSSGIUKWMPK
|
7.0 | IC50 | 2 | — | |
KRDDFKSJWNNSAT
|
7.0 | IC50 | 3 | — | |
LSJWYMSFUWBGPN
|
7.0 | IC50 | 17 | — | |
LVTITHFSOZBRMM
|
7.0 | IC50 | 2 | — | |
MBUVEWMHONZEQD
|
7.0 | IC50 | 17 | Yes | |
MJSCITFSPOLAGH
|
7.0 | IC50 | 3 | — | |
OCSZOZIYXZJENV
|
7.0 | IC50 | 3 | — | |
OHODDACZFUFQDV
|
7.0 | IC50 | 7 | — | |
OVTAMJUJNVINGX
|
7.0 | IC50 | 2 | — | |
PFSGEFYLEHABKV
|
7.0 | IC50 | 3 | — | |
SIKKESBUGBWVRF
|
7.0 | IC50 | 3 | — | |
SIYLLGKDQZGJHK
|
7.0 | IC50 | 13 | — | |
UYNVMODNBIQBMV
|
7.0 | IC50 | 10 | — | |
UYNVMODNBIQBMV
|
7.0 | IC50 | 5 | — | |
VFBZQFVDFIBXGZ
|
7.0 | Ki | 3 | — | |
VRZIEXXJAZACPZ
|
7.0 | IC50 | 7 | — | |
WOSGPVNODROINW
|
7.0 | IC50 | 2 | — | |
WUCNLBAXCJABQR
|
7.0 | IC50 | 2 | — | |
XQAYTEUNMDESNV
|
7.0 | Ki | 5 | — | |
YSWYESAJMAXMOW
|
7.0 | IC50 | 2 | — | |
YXISLLAVLYFJLK
|
7.0 | IC50 | 2 | — | |
YYYWTXUDIDHHTH
|
7.0 | Ki | 2 | — | |
ZUJPXZIUFHGAJI
|
7.0 | Ki | 3 | — | |
TVKCCIBAUDHHBL
|
7.0 | Ki | 2 | — | |
DQUUMUHVZGIZNI
|
7.0 | Ki | 2 | — | |
FIDXYKFRGLNFAF
|
7.0 | IC50 | 2 | — | |
SHNNJOOHYANVQG
|
7.0 | IC50 | 2 | — | |
FWSGJSPLQMXYQA
|
7.0 | Ki | 2 | — | |
GFZFUQFFPIRNGH
|
7.0 | IC50 | 2 | — | |
HMDHSUIMQILHRP
|
7.0 | Ki | 4 | — | |
IWFOFMOHDIUVDV
|
7.0 | IC50 | 2 | — | |
NNHSFUJHEDZYGF
|
7.0 | IC50 | 2 | — | |
SLYBJCUKCICSBD
|
7.0 | IC50 | 4 | Yes | |
UUEDQZRCAVWNIH
|
7.0 | IC50 | 2 | — | |
XWGNKABGVNJFEL
|
7.0 | Ki | 2 | — | |
XWGNKABGVNJFEL
|
7.0 | Ki | 2 | — | |
KDMBMLINAPXLCW
|
7.0 | IC50 | 3 | — | |
SNBBROUTMGTRAU
|
7.0 | Ki | 2 | — | |
LFSBNTMFCXGIEC
|
6.9 | Ki | 2 | — | |
XFUXIQVTGGYUOZ
|
6.9 | IC50 | 2 | — | |
ALWYLDGQXRIBHM
|
6.9 | IC50 | 2 | — | |
KGFPROOGUUWDFD
|
6.9 | IC50 | 2 | — | |
NMEPMLDUQJFQOK
|
6.9 | IC50 | 3 | — | |
NRKLSKYRBUUDLU
|
6.9 | Ki | 3 | — | |
SDFXSBFOVNINTE
|
6.9 | IC50 | 2 | — | |
TUISOQBOQRFWFJ
|
6.9 | Ki | 2 | — | |
XCFWDLWOCXSJOK
|
6.9 | IC50 | 2 | — | |
YEHCICAEULNIGD
|
6.9 | IC50 | 20 | — | |
PQWWHNZAZANFOZ
|
6.9 | IC50 | 5 | — | |
BLQLPPFWAKBJSW
|
6.9 | IC50 | 3 | — |