Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AXPVGJNPJSMCLA
|
7.2 | IC50 | 2 | — | |
ILIWVAFIMXCJTB
|
7.2 | Ki | 2 | — | |
MXXYXEAKIQRROV
|
7.2 | Ki | 4 | — | |
AVFYUSOOXDDQAW
|
7.1 | Ki | 2 | — | |
KCCUYRWFHHFONN
|
7.1 | IC50 | 2 | — | |
QCBWHGJPALSFJR
|
7.1 | Ki | 2 | — | |
YRRXDGSRIMGDFU
|
7.1 | IC50 | 2 | — | |
YIJMYSUOYUNZGL
|
7.1 | IC50 | 4 | — | |
ZBUMCITULAAXBQ
|
7.1 | Ki | 4 | — | |
DEIXGWIQADAVTO
|
7.1 | IC50 | 3 | — | |
DFXJFEAHWLUMQK
|
7.1 | IC50 | 3 | — | |
FNTHJTUPRVAXFZ
|
7.1 | IC50 | 17 | — | |
GESNZTWIXMSIMZ
|
7.1 | IC50 | 3 | — | |
HXGBXQDTNZMWGS
|
7.1 | IC50 | 8 | — | |
MCGIWMYXNXWIGG
|
7.1 | IC50 | 2 | — | |
MIHZNEWRGNWDAZ
|
7.1 | IC50 | 2 | — | |
MONKRYYJEIHBRU
|
7.1 | Ki | 4 | — | |
QDNROJXIPJKYJU
|
7.1 | Ki | 2 | — | |
QWKZREQFPCVBBG
|
7.1 | IC50 | 2 | — | |
TYDNACGHSINKSF
|
7.1 | Ki | 2 | — | |
UXQVMDVKHFQOEU
|
7.1 | IC50 | 5 | — | |
VNSQNNPGGZXQAN
|
7.1 | IC50 | 4 | — | |
XQNZVPNZMRIJKI
|
7.1 | IC50 | 2 | — | |
MVPXMHNFAQUXRM
|
7.1 | IC50 | 2 | — | |
RGZNEXHZUKHBNS
|
7.1 | IC50 | 2 | — | |
ULEWURLSYSOHEP
|
7.1 | IC50 | 3 | — | |
JKQCQYBXDQPJNC
|
7.1 | Ki | 3 | — | |
SRLHPXQPUSGNLH
|
7.1 | IC50 | 2 | — | |
PKQRYUSYILGVOB
|
7.1 | IC50 | 2 | — | |
QTQRWXSELPXXAV
|
7.1 | IC50 | 2 | — | |
SHCFFLWIRMAQPN
|
7.1 | Ki | 2 | — | |
IDHCWOUPGCDUGN
|
7.0 | Ki | 2 | — | |
WZSXQZNHMKLIIQ
|
7.0 | Ki | 2 | — | |
XCCMZNKLKPVPJT
|
7.0 | Ki | 2 | — | |
GMCICJZIANWTML
|
7.0 | IC50 | 2 | — | |
JEQFZUJUYZOZAL
|
7.0 | IC50 | 2 | — | |
RPPOAMDDJXHPIC
|
7.0 | IC50 | 2 | — | |
NCFNOILQWULHEZ
|
7.0 | Ki | 2 | — | |
BFEIADQANSGVFP
|
7.0 | IC50 | 2 | — | |
MCMNYTOHUPZLOA
|
7.0 | IC50 | 5 | — | |
BEXPSWDCLXOHKK
|
7.0 | Ki | 3 | — | |
FHRUVVOXWGOVFG
|
7.0 | Ki | 2 | — | |
APZHXGIRWMPKDR
|
7.0 | IC50 | 3 | — | |
FVBRGBXYCPMCNB
|
7.0 | IC50 | 3 | — | |
GIZYIOOBBUHOBS
|
7.0 | IC50 | 3 | — | |
HJLCHLAAXMALNR
|
7.0 | IC50 | 2 | — | |
HJWWNWMERDPVMY
|
7.0 | IC50 | 3 | — | |
HRUTWQCXFHLYSD
|
7.0 | IC50 | 2 | — | |
IVXOADYRPYSQPC
|
7.0 | IC50 | 3 | — | |
KEJJLAINBBOGHE
|
7.0 | IC50 | 2 | — |