Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OJZXUFDBDMQATJ
|
7.4 | IC50 | 4 | — | |
PIYDNEWDZZFKKO
|
7.4 | Ki | 2 | — | |
WNRRQSNNNIIUDN
|
7.4 | Ki | 3 | — | |
ZNGLHHGXOQHVRP
|
7.4 | IC50 | 2 | — | |
LKUBJXGOOGUQGP
|
7.4 | Ki | 2 | — | |
ITEQLSGAAAJLOU
|
7.4 | IC50 | 2 | — | |
MPQQLIGMXDXMJD
|
7.4 | Ki | 2 | — | |
ILPQLCKGOBBIPI
|
7.3 | IC50 | 2 | — | |
OGKTZPPCIHRDMM
|
7.3 | Ki | 2 | — | |
OOGJQPCLVADCPB
|
7.3 | IC50 | 9 | — | |
BHEGDYSAYYZJGP
|
7.3 | IC50 | 2 | — | |
QCLXNOBXQUWUEW
|
7.3 | IC50 | 9 | — | |
JIYPGFPFAVEPFX
|
7.3 | IC50 | 2 | — | |
RMQURPVWFQWESL
|
7.3 | Ki | 2 | — | |
ZJMZNFQDSWTHLP
|
7.3 | IC50 | 2 | — | |
ANYPUOSSIOCSJC
|
7.3 | IC50 | 3 | — | |
NHDILTZHICULAX
|
7.3 | Ki | 10 | — | |
PTVITZRFRXZZEA
|
7.3 | IC50 | 4 | — | |
VFIDGXZRONKQBZ
|
7.3 | IC50 | 5 | — | |
YANGEESWIGIKOP
|
7.3 | IC50 | 7 | Yes | |
GHTORLCXAYWNJL
|
7.3 | IC50 | 2 | — | |
QXIJKQBZACKAMG
|
7.3 | IC50 | 2 | — | |
JEUSLIAZMCQUCV
|
7.3 | IC50 | 2 | — | |
RWPWIJKKWCFKJJ
|
7.3 | IC50 | 2 | — | |
GGPDSNHLDADOIF
|
7.2 | IC50 | 2 | — | |
NIAOMAGQEARZHM
|
7.2 | IC50 | 2 | — | |
OUDYUUVZVNMOPP
|
7.2 | Ki | 3 | — | |
BDJJZYXDJQVPIV
|
7.2 | IC50 | 2 | — | |
DDHSIUUOIYFUOU
|
7.2 | Ki | 2 | — | |
KLBQZWRITKRQQV
|
7.2 | IC50 | 25 | Yes | |
XPWLJXVUAOISOS
|
7.2 | IC50 | 3 | — | |
AKZKUGUQZMUCJC
|
7.2 | IC50 | 2 | — | |
JFLFBSAQNKZEKC
|
7.2 | IC50 | 2 | — | |
OKRHAYBIIRGRNK
|
7.2 | IC50 | 2 | — | |
PDKGFOSJNKVHSS
|
7.2 | IC50 | 2 | — | |
PRAXUIQVVJSJMP
|
7.2 | Ki | 2 | — | |
ADHCEOHLWFBYCU
|
7.2 | Ki | 2 | — | |
JGRNPFVRYKMKOL
|
7.2 | IC50 | 2 | — | |
IMFBORACXDJQCD
|
7.2 | IC50 | 3 | — | |
KGVROJQOCQABGA
|
7.2 | Ki | 7 | — | |
MMHPZQOEUVHNBB
|
7.2 | IC50 | 3 | — | |
NNCTXKNNQUMOPC
|
7.2 | IC50 | 3 | — | |
OVGUUSWJYHCFLN
|
7.2 | IC50 | 3 | — | |
SAMYTBZVLLYSKN
|
7.2 | IC50 | 5 | — | |
VLAMSHNLMPNZGJ
|
7.2 | IC50 | 2 | — | |
VVYQHHROMNFSAO
|
7.2 | IC50 | 4 | — | |
IFFPICMESYHZPQ
|
7.2 | IC50 | 4 | — | |
GXZNBYLIQYWZLV
|
7.2 | IC50 | 2 | — | |
LCQVKIHGMHPFIJ
|
7.2 | IC50 | 2 | — | |
RTHCYVBBDHJXIQ
|
7.2 | IC50 | 15 | — |