Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LOGDXDWDCZTLOS
|
7.6 | IC50 | 3 | — | |
SEWIXNYQXNASBQ
|
7.6 | IC50 | 2 | — | |
SKGSBVPKDPLIEF
|
7.6 | Ki | 5 | — | |
YGDMWGYWZVBWDP
|
7.6 | IC50 | 3 | — | |
FDZFVXKCJKOSRC
|
7.6 | IC50 | 2 | — | |
SCAVCNGNYHPFKS
|
7.6 | Ki | 2 | — | |
YLSHULIHKQRKEM
|
7.6 | IC50 | 4 | — | |
WYHMARFYRUASMT
|
7.6 | IC50 | 2 | — | |
XYUYSDBKGVJSKN
|
7.6 | IC50 | 5 | — | |
SPZVGUOPAIQFIW
|
7.5 | IC50 | 2 | — | |
VSACRBUHJYUONF
|
7.5 | IC50 | 2 | — | |
BHWGZPATDOVSCG
|
7.5 | IC50 | 2 | — | |
CVUXESFCUHCXHB
|
7.5 | IC50 | 2 | — | |
CZXRKQNLGWTZPP
|
7.5 | IC50 | 2 | — | |
FXUCYRRIEXLTRF
|
7.5 | IC50 | 2 | — | |
IAFSRSYSLPAOJE
|
7.5 | IC50 | 2 | — | |
LNEPOXFFQSENCJ
|
7.5 | IC50 | 33 | Yes | |
ZGQXJAMXZIFYHC
|
7.5 | Ki | 2 | — | |
DPAGUJADGMJVKD
|
7.5 | Ki | 5 | — | |
GPZNPXAPAFLRLB
|
7.5 | IC50 | 2 | — | |
KQTXWKJKIOAAAJ
|
7.5 | IC50 | 2 | — | |
UGDQKRGYVYUTTP
|
7.5 | Ki | 2 | — | |
WWTXVMIWFBVHQA
|
7.5 | IC50 | 2 | — | |
DAFKTUHZZXUBLN
|
7.5 | IC50 | 2 | — | |
CQOJHAJWCDJEAT
|
7.5 | IC50 | 3 | — | |
SGLJPXQOJMBPBR
|
7.5 | IC50 | 3 | — | |
RMEDXOLNCUSCGS
|
7.5 | IC50 | 17 | Yes | |
BKMZXLKUUMOTKA
|
7.5 | IC50 | 3 | — | |
RDOIQAHITMMDAJ
|
7.5 | IC50 | 13 | — | |
MVMGNWUSDKNEKN
|
7.5 | Ki | 5 | — | |
RZFIMUGJIHXZIF
|
7.5 | IC50 | 2 | — | |
GYVLPHYAFKCJIG
|
7.5 | Ki | 4 | — | |
XBIPCIFARHCNNE
|
7.5 | Ki | 4 | — | |
ALLIMXLDTJFWHR
|
7.4 | IC50 | 2 | — | |
AZGZXUZMWKHDDH
|
7.4 | IC50 | 2 | — | |
DCSUBABJRXZOMT
|
7.4 | IC50 | 2 | — | |
PPLVDBKGJPKXLH
|
7.4 | IC50 | 4 | — | |
SXFCZOCWXLILSQ
|
7.4 | IC50 | 2 | — | |
AXXCMOIEGOZRPQ
|
7.4 | IC50 | 2 | — | |
DDNCQMVWWZOMLN
|
7.4 | IC50 | 2 | — | |
ULGZDMOVFRHVEP
|
7.4 | IC50 | 59 | — | |
DCSUBABJRXZOMT
|
7.4 | IC50 | 24 | — | |
FLZIWHXEHDCVMN
|
7.4 | Ki | 2 | — | |
HMXWHDMFAKYACA
|
7.4 | IC50 | 3 | — | |
MPCLARAFXPQZQF
|
7.4 | IC50 | 2 | — | |
OZUYIQYXHKJSCF
|
7.4 | IC50 | 4 | — | |
PKAXIMFUJIQFKS
|
7.4 | IC50 | 3 | — | |
URTQOVWDFKPXTI
|
7.4 | IC50 | 3 | — | |
VBQPFBIQLMTMNM
|
7.4 | IC50 | 3 | — | |
LKRTVYMJTLSROG
|
7.4 | Ki | 2 | — |