Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZFSIPUPFUSVPMQ
|
7.8 | IC50 | 2 | — | |
ZFSIPUPFUSVPMQ
|
7.8 | IC50 | 2 | — | |
RASPHJGGIPBIMT
|
7.8 | IC50 | 2 | — | |
FLLIMXCHPPVPAF
|
7.8 | IC50 | 3 | — | |
FVFURMJFTAJXRH
|
7.8 | IC50 | 3 | — | |
MTFGAWDMZPCQKM
|
7.8 | IC50 | 2 | — | |
FQXDXSUCYIDGPA
|
7.8 | IC50 | 2 | — | |
IBVNIPPBTCWYJG
|
7.8 | IC50 | 2 | — | |
KESABOVUGAHUQM
|
7.8 | IC50 | 2 | — | |
LLWKBGRAWPNWFD
|
7.8 | IC50 | 2 | — | |
LNKQLDXMYFJALH
|
7.8 | Ki | 2 | — | |
MAVYUWKKUQUUJD
|
7.8 | IC50 | 2 | — | |
YEQFSCLZXBNXBX
|
7.8 | IC50 | 2 | — | |
YZAHEHXQIMZHAJ
|
7.8 | IC50 | 5 | — | |
ZBIAKUMOEKILTF
|
7.8 | IC50 | 2 | — | |
BHWGZPATDOVSCG
|
7.8 | IC50 | 2 | — | |
MWIXMEAIQGTQEO
|
7.8 | IC50 | 2 | — | |
RQQJZPUPHSLLRR
|
7.8 | IC50 | 2 | — | |
RRZYXZCEHAPBIS
|
7.8 | IC50 | 2 | — | |
LZZYJVMGDLEHFH
|
7.8 | IC50 | 2 | — | |
QOUVFTQPYVSKEQ
|
7.8 | Ki | 4 | — | |
RMHSPVDIAHEXNT
|
7.8 | IC50 | 2 | — | |
SBFDBMKEWKLRSB
|
7.8 | IC50 | 2 | — | |
CSPMIMZHBXUYLQ
|
7.7 | Ki | 2 | — | |
NZGLSOKQCCNTMG
|
7.7 | IC50 | 2 | — | |
QSCBMVHTDSJVEE
|
7.7 | IC50 | 3 | — | |
WFZUDDFKDDQSCZ
|
7.7 | IC50 | 2 | — | |
OHLDJJXRTLZQSU
|
7.7 | IC50 | 3 | — | |
COLOFELGEFWPSM
|
7.7 | IC50 | 2 | — | |
FEQJNVMOFHFOGP
|
7.7 | IC50 | 3 | — | |
ITLZCAFYUUBRFV
|
7.7 | IC50 | 2 | — | |
MIVZTSHUBPAZML
|
7.7 | IC50 | 3 | — | |
ORRBREIXBAIZTQ
|
7.7 | Ki | 4 | — | |
WCNMMPUKVKKLKP
|
7.7 | IC50 | 2 | — | |
YJAIZWWQRYKSON
|
7.7 | IC50 | 2 | — | |
YVUQSNJEYSNKRX
|
7.7 | IC50 | 36 | — | |
ZZCFQOGPJUCWRJ
|
7.7 | IC50 | 2 | — | |
GQQMDOGXIJRPDK
|
7.7 | IC50 | 2 | — | |
IRDUJBOZWQOVPG
|
7.7 | IC50 | 2 | — | |
YECSPBDBORKKPX
|
7.7 | IC50 | 2 | — | |
VRUSWBLOISBSSJ
|
7.7 | IC50 | 5 | — | |
AFZGUFJUAJQREI
|
7.6 | IC50 | 2 | — | |
KTRMFSXYMXPKHJ
|
7.6 | IC50 | 2 | — | |
XZEWWPFRVAGHEH
|
7.6 | IC50 | 2 | — | |
IZVROLMEXNRNHZ
|
7.6 | IC50 | 4 | Yes | |
JFJGUHDHENWREH
|
7.6 | IC50 | 2 | — | |
OKLKDPLBWBNFAN
|
7.6 | IC50 | 2 | — | |
PZUJQWHTIRWCID
|
7.6 | IC50 | 7 | — | |
HZNTWQAMIOKCMC
|
7.6 | IC50 | 2 | — | |
IYEJAIHDFCXVRY
|
7.6 | IC50 | 2 | — |