Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BZNSXKFFBJLSJV
|
8.1 | IC50 | 2 | — | |
RCSMYQHGJMPVOW
|
8.1 | IC50 | 2 | — | |
WQIJWPZIOIFLHO
|
8.1 | IC50 | 2 | — | |
YUMXUYVBLHCRQN
|
8.1 | IC50 | 2 | — | |
MRUYVXJFVOSZEV
|
8.1 | IC50 | 2 | — | |
AYNOFJPXPRZEFF
|
8.1 | IC50 | 2 | — | |
NKKHUNXEXXFYQF
|
8.1 | IC50 | 2 | — | |
AMRUTRWUTNIKQI
|
8.1 | IC50 | 2 | — | |
QVUDEDBAGYAVHI
|
8.1 | IC50 | 2 | — | |
YZMMWVWLDOCLCK
|
8.1 | IC50 | 2 | — | |
ZZFKFTVPUSBMNB
|
8.1 | IC50 | 2 | — | |
ANCFKYJMXNMYNZ
|
8.1 | IC50 | 3 | — | |
VQGLUTISKQTZKB
|
8.1 | IC50 | 2 | — | |
WPSWNDSKLXFMIS
|
8.1 | IC50 | 2 | — | |
XPWXBGYLYLSHTG
|
8.1 | IC50 | 2 | — | |
JTXZPQNLRJKZDT
|
8.0 | IC50 | 2 | — | |
CIHRMKSTNVZPFD
|
8.0 | IC50 | 2 | — | |
RVVNCNQGXBSLJG
|
8.0 | IC50 | 2 | — | |
BZUVXLPHVGFEJA
|
8.0 | IC50 | 2 | — | |
WYHMARFYRUASMT
|
8.0 | IC50 | 2 | — | |
AMJYDFFNPACSTJ
|
8.0 | IC50 | 2 | — | |
KFOXMHFDNRTETJ
|
8.0 | Ki | 5 | — | |
KVVCXQIQAOOKFF
|
8.0 | IC50 | 3 | — | |
VVGHIMUWASPVQJ
|
8.0 | IC50 | 3 | — | |
WSEQXVZVJXJVFP
|
8.0 | IC50 | 6 | Yes | |
AIDALYBWFLHEJP
|
8.0 | IC50 | 2 | — | |
PGRNXALRNBGGDQ
|
8.0 | IC50 | 2 | — | |
AOIKKLIBKSSHQP
|
8.0 | Ki | 4 | — | |
DOAPNMVLEGQTQO
|
8.0 | IC50 | 2 | — | |
YYOXBGHALUHPAP
|
8.0 | IC50 | 2 | — | |
BLVUILRZDGFJPZ
|
7.9 | IC50 | 2 | — | |
AIPQYPCEXRVEFE
|
7.9 | IC50 | 2 | — | |
BYNZSRRNMOCSHJ
|
7.9 | IC50 | 2 | — | |
GAXRSLAUXVLRCM
|
7.9 | IC50 | 2 | — | |
NTFKMMZGMLEXET
|
7.9 | IC50 | 2 | — | |
PBDMWGSHTOZGOM
|
7.9 | IC50 | 6 | — | |
RIDRYHZYVUEBMC
|
7.9 | IC50 | 2 | — | |
UMQXZSKUBTWYIX
|
7.9 | IC50 | 2 | — | |
HZEJTMIZKGGUNU
|
7.9 | IC50 | 2 | — | |
UDROTHQORZMMBF
|
7.9 | IC50 | 2 | — | |
COVZSEBDZICBKI
|
7.9 | IC50 | 2 | — | |
FBZSCRZWBGBTTM
|
7.9 | Ki | 2 | — | |
GQQMDOGXIJRPDK
|
7.9 | IC50 | 2 | — | |
IDPGDKXBQTZRGW
|
7.9 | IC50 | 2 | — | |
JFHIYLBDXQPCLD
|
7.9 | IC50 | 2 | — | |
MHZCWVOMNJUVMC
|
7.9 | IC50 | 2 | — | |
FNMSKRVJSVGVRH
|
7.8 | Ki | 2 | — | |
GZKLJWGUPQBVJQ
|
7.8 | IC50 | 24 | Yes | |
QQKFLUBSTABOJV
|
7.8 | Ki | 3 | — | |
WKBMRZDYCZPLFO
|
7.8 | IC50 | 6 | — |