Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AMZHEQZGCLSTMF
|
8.3 | IC50 | 2 | — | |
HZNTWQAMIOKCMC
|
8.3 | IC50 | 2 | — | |
ITQFRPBHRRDOKY
|
8.3 | IC50 | 3 | — | |
NTFKMMZGMLEXET
|
8.3 | IC50 | 2 | — | |
PVFFECNHTDFMJH
|
8.3 | IC50 | 3 | — | |
SJTLVMWWYORGEH
|
8.3 | Ki | 2 | — | |
UJXZIZJAELMUHW
|
8.3 | Ki | 2 | — | |
VJPTYAZXVBTBPT
|
8.3 | IC50 | 2 | — | |
JYOPFNFGXYLUHA
|
8.3 | Ki | 2 | — | |
WXODWEUHUBMNAU
|
8.3 | IC50 | 2 | — | |
WXIFVEVHNGMUHP
|
8.3 | IC50 | 2 | — | |
MZNNAIHCWWROJM
|
8.3 | IC50 | 2 | — | |
PQZGPKXZUSHGLE
|
8.2 | IC50 | 2 | — | |
UGWKDYRCSUMLFR
|
8.2 | IC50 | 2 | — | |
BZFJGKHIEZMTSV
|
8.2 | Ki | 2 | — | |
JUMJODAYGHYIAH
|
8.2 | IC50 | 2 | — | |
KTNRAOBLSVMKID
|
8.2 | IC50 | 2 | — | |
LOVAEQYMKDVCHF
|
8.2 | IC50 | 2 | — | |
UEPQDBDTOSJGSX
|
8.2 | IC50 | 2 | — | |
URGBLKJMXGEIKS
|
8.2 | IC50 | 2 | — | |
WFZUDDFKDDQSCZ
|
8.2 | IC50 | 2 | — | |
FTOGLQXKLWNGLW
|
8.2 | Ki | 2 | — | |
GXDALQBWZGODGZ
|
8.2 | IC50 | 21 | Yes | |
IDPGDKXBQTZRGW
|
8.2 | IC50 | 2 | — | |
UAFYSVAOAUUNBN
|
8.2 | IC50 | 3 | — | |
KWGHMJGFVYVORH
|
8.2 | IC50 | 2 | — | |
LXPLSZAVQYCVGQ
|
8.2 | IC50 | 2 | — | |
JQEQULOLEPTBRS
|
8.2 | IC50 | 3 | — | |
CSMSBZWRUZAKQB
|
8.2 | IC50 | 2 | — | |
PHBYNJGKPFJBPE
|
8.2 | IC50 | 2 | — | |
MXAUIAYYRYRHPY
|
8.2 | Ki | 2 | — | |
VJISUJZHUGWEPY
|
8.2 | IC50 | 3 | — | |
IZLJKNPYMLZCPG
|
8.2 | IC50 | 2 | — | |
MULJMOFCKZZSRK
|
8.2 | IC50 | 2 | — | |
MKAPFCBLWCECBI
|
8.2 | IC50 | 2 | — | |
RJVPOCVCIFLEDC
|
8.2 | IC50 | 2 | — | |
CIMJGOFPRRZLKM
|
8.2 | IC50 | 2 | — | |
GKZBQPSXHBJOPU
|
8.2 | IC50 | 2 | — | |
NVDMYRPSMBTQKR
|
8.2 | IC50 | 2 | — | |
SJLQMBIPYINRMF
|
8.2 | IC50 | 2 | — | |
CYBJAJOVKOECGI
|
8.1 | IC50 | 2 | — | |
KBSGBIFMBKBFMH
|
8.1 | IC50 | 2 | — | |
QCQXHPGCLHGFID
|
8.1 | IC50 | 2 | — | |
DOYKZJFYZSSDTP
|
8.1 | IC50 | 2 | — | |
GHQQXFVYIYQRDG
|
8.1 | IC50 | 2 | — | |
CQIHYFQHPBTXLQ
|
8.1 | Ki | 2 | — | |
LHMLJRCNGQZNHL
|
8.1 | IC50 | 2 | — | |
MJOSWDSZKHMYMF
|
8.1 | Ki | 2 | — | |
NCDNWTYTZTXJIU
|
8.1 | IC50 | 3 | — | |
YUBLNBWIZGHBST
|
8.1 | IC50 | 2 | — |