Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PBTFDTKJUCHOCI
|
8.7 | IC50 | 2 | — | |
HPMOYSAWXGTKNO
|
8.6 | IC50 | 2 | — | |
IYVIYWIRAJCIRW
|
8.6 | IC50 | 2 | — | |
FVIRTVGXWNRAMY
|
8.6 | IC50 | 2 | — | |
YHVMAQQCYJWINX
|
8.6 | IC50 | 2 | — | |
PPMFNADUOOVZPG
|
8.6 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
8.6 | IC50 | 165 | Yes | |
ICFZXEQTLNSVSO
|
8.6 | IC50 | 2 | — | |
BFXKWHZHXIVGOE
|
8.6 | IC50 | 2 | — | |
FWWHNGKEZAFESY
|
8.6 | IC50 | 2 | — | |
RMNBHDPKKIBKOP
|
8.6 | IC50 | 2 | — | |
YFSPDWGKSWOSRI
|
8.6 | IC50 | 2 | — | |
LEHFCHSREMRJMI
|
8.5 | IC50 | 2 | — | |
QIMVRHMVKAJIDE
|
8.5 | IC50 | 2 | — | |
RRRMNLLTGSQHGV
|
8.5 | IC50 | 2 | — | |
DJTVQVIZMNHBCR
|
8.5 | IC50 | 2 | — | |
FFCXAJUMJUOFPK
|
8.5 | IC50 | 2 | — | |
IIXUBHOQXODODU
|
8.5 | IC50 | 3 | — | |
NEBCCMOWOJKFFS
|
8.5 | IC50 | 3 | — | |
UDHXHJAZPMOTOA
|
8.5 | IC50 | 3 | — | |
XNQLYGHTCMOZRQ
|
8.5 | IC50 | 3 | — | |
GQOXXKSNEOMYOB
|
8.5 | IC50 | 2 | — | |
WJNQZXPCJCLCNG
|
8.5 | IC50 | 6 | — | |
DMCNIEIKHCMYAH
|
8.5 | IC50 | 2 | — | |
NNKIFQRRDDJHKS
|
8.5 | IC50 | 2 | — | |
NEVDMWBUYBQSHQ
|
8.5 | IC50 | 2 | — | |
HJXJZSZXJNHUQH
|
8.4 | IC50 | 2 | — | |
SADTVAAIAQIVQH
|
8.4 | IC50 | 2 | — | |
SWOGBCMCJSXRTN
|
8.4 | IC50 | 2 | — | |
FDUQYLYBWZAWAD
|
8.4 | IC50 | 2 | — | |
ICIUVKVSEXZBQM
|
8.4 | IC50 | 2 | — | |
OBNOGIWVGBFGEH
|
8.4 | IC50 | 2 | — | |
SFKBOTCVPFRCEE
|
8.4 | IC50 | 2 | — | |
FNEORDYLRZOEEP
|
8.4 | IC50 | 5 | — | |
GDXMDKRKEIKPLW
|
8.4 | IC50 | 3 | — | |
HHCYCBKPWYJVEB
|
8.4 | IC50 | 3 | — | |
HNONCNSCKGVMAR
|
8.4 | IC50 | 2 | — | |
KETIMUXEJZGZHT
|
8.4 | IC50 | 2 | — | |
LCCYGLSQPCXNFG
|
8.4 | IC50 | 2 | — | |
SNGNEJSZIKADBS
|
8.4 | IC50 | 2 | — | |
SNGNEJSZIKADBS
|
8.4 | IC50 | 2 | — | |
GJOARULBWVWENP
|
8.4 | IC50 | 2 | — | |
YHMGBTHOLTYBSS
|
8.4 | IC50 | 2 | — | |
DREYZGCIOLBBDK
|
8.4 | IC50 | 2 | — | |
ZPUCINDJVBIVPJ
|
8.4 | IC50 | 4 | — | |
VAHPGMWAHQHAMJ
|
8.3 | IC50 | 2 | — | |
CSQOOKHGXFRBEQ
|
8.3 | Ki | 2 | — | |
RJVPOCVCIFLEDC
|
8.3 | IC50 | 2 | — | |
WLLRAGBPCSOJNH
|
8.3 | Ki | 2 | — | |
IQTXUDCVFFYTOM
|
8.3 | IC50 | 2 | — |