Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WLWQLJYOYMGFPD
|
6.4 | IC50 | 2 | — | |
XQRZVIKHJWAVPW
|
6.4 | IC50 | 2 | — | |
AFUIBDRITZEBAF
|
6.4 | Ki | 2 | — | |
FYIAXSYXQPAMIK
|
6.4 | IC50 | 7 | — | |
PNOVIOUSABCJCS
|
6.4 | IC50 | 3 | — | |
PYKXSNLYPSZMTQ
|
6.4 | IC50 | 4 | — | |
QSFGBNSTSAEDNQ
|
6.4 | IC50 | 2 | — | |
SUBIMNIDAXOLTK
|
6.4 | IC50 | 7 | — | |
ULRYFJLRJZVHIZ
|
6.4 | IC50 | 7 | — | |
WHGLFZPJAYDODK
|
6.4 | IC50 | 3 | — | |
WUANGOCWSCYKOJ
|
6.4 | IC50 | 2 | — | |
AIBNCLLVENCCGP
|
6.4 | IC50 | 2 | — | |
AJBBNBBBDUCRTB
|
6.4 | IC50 | 2 | — | |
AMOACTSTZUXXDX
|
6.4 | IC50 | 4 | — | |
ASRDPULQBHFPGU
|
6.4 | IC50 | 7 | — | |
BILQJDKHRSUCQZ
|
6.4 | Ki | 5 | — | |
BNDVRMMWXZWPSL
|
6.4 | IC50 | 2 | — | |
BTFVTAWVFBWGHC
|
6.4 | IC50 | 4 | — | |
BXZGSIDSJSGAJE
|
6.4 | IC50 | 2 | — | |
CGMNUBKHKAKYOW
|
6.4 | Ki | 2 | — | |
CNMDDAFIBJNBFQ
|
6.4 | Ki | 2 | — | |
CXDMEJPMIGCWHH
|
6.4 | Ki | 2 | — | |
DXWFZCDHFLBXON
|
6.4 | IC50 | 2 | — | |
GJJQUHQSJVEHNN
|
6.4 | IC50 | 2 | — | |
HEHHNIMMUJHLIO
|
6.4 | Ki | 5 | — | |
HFXUYZQVCSUBMO
|
6.4 | Ki | 2 | — | |
IKHRYIGPRIAKFA
|
6.4 | IC50 | 3 | — | |
JGRQIRDAIIUUCX
|
6.4 | IC50 | 3 | — | |
JJKMOFKIYHXREY
|
6.4 | IC50 | 5 | — | |
KBYDKOYJEQUBOE
|
6.4 | IC50 | 2 | — | |
KFCVKULFYARZLT
|
6.4 | IC50 | 2 | — | |
KFHYZKCRXNRKRC
|
6.4 | Ki | 2 | — | |
KONPIFGGWNMOKY
|
6.4 | IC50 | 4 | — | |
LHNFCNUXICTTPA
|
6.4 | IC50 | 2 | — | |
LSPPODQSTNTKTE
|
6.4 | IC50 | 2 | — | |
LXGZSTDLYCGLAE
|
6.4 | IC50 | 4 | — | |
MSXJZHUTIDWQBZ
|
6.4 | IC50 | 8 | — | |
MVXIVGJQLGJBTD
|
6.4 | Ki | 2 | — | |
NCLSCERPSPVBHT
|
6.4 | IC50 | 2 | — | |
OMOJVKDXKKEFQT
|
6.4 | IC50 | 3 | — | |
OOZRFFVYRKXFKQ
|
6.4 | IC50 | 2 | — | |
OZOLNJQERDKPFN
|
6.4 | IC50 | 2 | — | |
OZOLNJQERDKPFN
|
6.4 | IC50 | 2 | — | |
QKGFAFCTWJXMJH
|
6.4 | Ki | 2 | — | |
RSVBTLSIVBWMNF
|
6.4 | IC50 | 3 | — | |
SXKNFGNGCSTXQU
|
6.4 | Ki | 2 | — | |
TYLUAGXHVPXCPL
|
6.4 | IC50 | 2 | — | |
UAVBPSVJXCTZOC
|
6.4 | IC50 | 3 | — | |
VANBZHNBQWYEMT
|
6.4 | IC50 | 3 | — | |
VFCNPRIWDSWJIG
|
6.4 | IC50 | 2 | — |