Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SLVMESMUVMCQIY
|
6.5 | IC50 | 14 | — | |
UEBNHTSMTQUOQB
|
6.5 | IC50 | 2 | — | |
WAEXFXRVDQXREF
|
6.5 | IC50 | 20 | Yes | |
XADCESSVHJOZHK
|
6.5 | IC50 | 4 | — | |
BKGOKPQNNKWLHW
|
6.5 | IC50 | 2 | — | |
GETROLYXSDDSDH
|
6.5 | IC50 | 2 | — | |
QXLYDXQRLPSIKM
|
6.5 | IC50 | 2 | — | |
CPMLYZUSUXTRIP
|
6.5 | IC50 | 3 | — | |
CRBTZFVQVOXBBO
|
6.5 | Ki | 2 | — | |
GTPUUTXWVUCADD
|
6.5 | Ki | 2 | — | |
GZNVXAZGAACUQD
|
6.5 | IC50 | 2 | — | |
JTOFILOVFYOIGD
|
6.5 | IC50 | 3 | — | |
VSHOBSIPZJJYRP
|
6.5 | IC50 | 2 | — | |
AWAWHJXFEZNWPV
|
6.5 | IC50 | 3 | — | |
IDTOXCSJPHTASJ
|
6.5 | IC50 | 2 | — | |
OBUQQSWVYWHDKA
|
6.5 | IC50 | 2 | — | |
ODIJMXCJWMOZFJ
|
6.5 | IC50 | 3 | — | |
OGHNVEJMJSYVRP
|
6.5 | IC50 | 18 | — | |
QMTPGEKECKOWFW
|
6.5 | IC50 | 2 | — | |
RDPSEAZFXPEZMP
|
6.5 | IC50 | 2 | — | |
WXZVOQCMUCSBIN
|
6.5 | IC50 | 3 | — | |
CXZDAMKDHUXFMW
|
6.5 | Ki | 4 | — | |
RMXXLBXAQDDMHW
|
6.5 | Ki | 2 | — | |
BCRSYZQXPRWUJQ
|
6.4 | IC50 | 3 | — | |
JZEQFVDLSUHIOP
|
6.4 | Ki | 2 | — | |
KHWFDRKDQCSBEW
|
6.4 | IC50 | 2 | — | |
LDCYRYGDVBLWLI
|
6.4 | IC50 | 2 | — | |
LVQKKHWEPPQIMP
|
6.4 | Ki | 2 | — | |
OGJWWUCDNHVDOY
|
6.4 | IC50 | 4 | — | |
OWMBYQVIMDTSAW
|
6.4 | IC50 | 2 | — | |
VBOXQXAJDAUESQ
|
6.4 | Ki | 2 | — | |
VMYIWPNMBCKTFR
|
6.4 | IC50 | 2 | — | |
ZEJPZPGMAWZAJD
|
6.4 | IC50 | 3 | — | |
CMMVRTXWYOGXHR
|
6.4 | IC50 | 4 | — | |
IHNSUBDSHNRLFA
|
6.4 | IC50 | 2 | — | |
KYASUVSAKOTGNF
|
6.4 | IC50 | 3 | — | |
MNAFRWGRFIBAQX
|
6.4 | IC50 | 3 | — | |
MQWFPEJVMZVZBQ
|
6.4 | Ki | 2 | — | |
QUIJNHUBAXPXFS
|
6.4 | IC50 | 2 | — | |
TZFKQPVOFBQHAZ
|
6.4 | IC50 | 9 | — | |
WLGVVEQIKFIUPU
|
6.4 | IC50 | 3 | — | |
CQVVMULTZQAZBA
|
6.4 | IC50 | 2 | — | |
FCVWUDUFOJNPPC
|
6.4 | IC50 | 2 | — | |
LETPPZNSGLCXSE
|
6.4 | IC50 | 3 | — | |
LWQXKZOHKORPRL
|
6.4 | IC50 | 2 | — | |
NABHHUMHJIHHIX
|
6.4 | IC50 | 4 | — | |
NFNUDBUGUZLOPA
|
6.4 | Ki | 2 | — | |
NYCIVVXGRDGDMY
|
6.4 | IC50 | 2 | — | |
SLKZDILCMYJAFM
|
6.4 | IC50 | 2 | — | |
SZALSWFXFHISRB
|
6.4 | Ki | 2 | — |