Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PPHJOGOEUDGEOR
|
6.5 | IC50 | 2 | — | |
PZWALEZJXWWGIX
|
6.5 | IC50 | 2 | — | |
QOOGOLVYWAKPMZ
|
6.5 | Ki | 2 | — | |
QUWFBAJQLUHXBF
|
6.5 | IC50 | 2 | — | |
RSVBTLSIVBWMNF
|
6.5 | IC50 | 3 | — | |
SDWQCOVERLZWAC
|
6.5 | Ki | 2 | — | |
UIZGWTRYQVFMHV
|
6.5 | Ki | 2 | — | |
UPKZNVQHJZHSGN
|
6.5 | Ki | 2 | — | |
VURLRACCOCGFDB
|
6.5 | IC50 | 6 | — | |
VVIXUMWNLIZSDM
|
6.5 | IC50 | 2 | — | |
WKNXCGCJMLOINR
|
6.5 | IC50 | 2 | — | |
YGUFCDOEKKVKJK
|
6.5 | Ki | 4 | — | |
YIXQZLPGNXXTFM
|
6.5 | IC50 | 2 | — | |
ZODXHEFTTJWNPK
|
6.5 | Ki | 3 | — | |
CFUPTNNNCZABDF
|
6.5 | IC50 | 2 | — | |
CKXRLZVQKNQKHJ
|
6.5 | IC50 | 4 | — | |
CNTAQWMENZCDOK
|
6.5 | IC50 | 2 | — | |
HKBQLXYNZOLAHS
|
6.5 | Ki | 2 | — | |
RWWMQYYGHIHOGU
|
6.5 | IC50 | 2 | — | |
RWZHKEZRFILBTQ
|
6.5 | IC50 | 2 | — | |
ANTOILZBKKIMIM
|
6.5 | IC50 | 2 | — | |
AUZMCSDTNJIOIN
|
6.5 | IC50 | 3 | — | |
CBWCJYFVVHOTAZ
|
6.5 | IC50 | 3 | — | |
CDPXETVZRHNLTM
|
6.5 | IC50 | 3 | — | |
CVUSIJVOABHLEJ
|
6.5 | Ki | 3 | — | |
FRYWDPTWXKMFIV
|
6.5 | IC50 | 3 | — | |
JYLNFWODPITKFP
|
6.5 | IC50 | 3 | — | |
KLQDZSYTMPJBBU
|
6.5 | IC50 | 3 | — | |
KOHIRBRYDXPAMZ
|
6.5 | IC50 | 2 | — | |
LCSARSYDEHXRBQ
|
6.5 | IC50 | 3 | — | |
LPHIWCBAJGQIIF
|
6.5 | IC50 | 3 | — | |
OACVKINMDRORAI
|
6.5 | IC50 | 3 | — | |
PQTUVUOTFUHROL
|
6.5 | Ki | 2 | — | |
QLOCSQXNJJSRQH
|
6.5 | IC50 | 3 | — | |
QRRCESJWXMIGPS
|
6.5 | IC50 | 2 | — | |
SINXEYLFXFHPMM
|
6.5 | Ki | 2 | — | |
SSMBSCUSIUNOPU
|
6.5 | IC50 | 3 | — | |
SXPUHRRIRIQRTP
|
6.5 | IC50 | 7 | — | |
SYOADIUGRJTHHU
|
6.5 | Ki | 8 | — | |
UOCMXNLGBQWJPG
|
6.5 | IC50 | 3 | — | |
VCJRZGBNXMAJCB
|
6.5 | IC50 | 2 | — | |
VSUKSHADZRDBII
|
6.5 | IC50 | 2 | — | |
XLJQOKQZCYRQNN
|
6.5 | IC50 | 3 | — | |
XUKSGYGUDPUQCB
|
6.5 | IC50 | 3 | — | |
YRAPNFDLJRSFKB
|
6.5 | Ki | 4 | — | |
YSDZQWRVRDWYHN
|
6.5 | Ki | 2 | — | |
ZOCPXKXAOXQZSF
|
6.5 | IC50 | 3 | — | |
LOUPRKONTZGTKE
|
6.5 | IC50 | 3 | — | |
MVXMOYOFQUJRHY
|
6.5 | Ki | 2 | — | |
QZUDBNBUXVUHMW
|
6.5 | IC50 | 39 | Yes |