Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GPDZHKOGLHALQL
|
6.6 | IC50 | 3 | — | |
KZTWANLURUNJBS
|
6.6 | Ki | 2 | — | |
AMLPUCGCCQQMBJ
|
6.6 | IC50 | 2 | — | |
BETCCFITWJNKCT
|
6.6 | Ki | 2 | — | |
CHLLVQZFMABVHW
|
6.6 | IC50 | 2 | — | |
FCYQRIODPYABJL
|
6.6 | IC50 | 3 | — | |
GOBNHYGEALNGCV
|
6.6 | IC50 | 3 | — | |
GPANICKLGIVBML
|
6.6 | Ki | 2 | — | |
OUUFVLURDMTSII
|
6.6 | Ki | 3 | — | |
RLHOWHVHHMGIKE
|
6.6 | IC50 | 3 | — | |
XBODCTVRQGLZFY
|
6.6 | IC50 | 2 | — | |
AXDZGPVPBMNCMT
|
6.6 | Ki | 4 | — | |
KVDPUCCGORKFOD
|
6.6 | Ki | 3 | — | |
PLOFBQMQAHOQHM
|
6.6 | Ki | 2 | — | |
NDCFZCPGTKKFMD
|
6.6 | Ki | 4 | — | |
CFUPTNNNCZABDF
|
6.5 | IC50 | 2 | — | |
COGCORROFSOJTQ
|
6.5 | IC50 | 3 | — | |
CXRCFQKCULIFAC
|
6.5 | Ki | 2 | — | |
DHCCENVMWQKDAG
|
6.5 | IC50 | 2 | — | |
JFKJLEGVSYQSFA
|
6.5 | Ki | 2 | — | |
SRVOWVHRVJSZKO
|
6.5 | IC50 | 3 | — | |
ULSSDVVGTBLGMG
|
6.5 | IC50 | 2 | — | |
AJNXRYLTABACFI
|
6.5 | IC50 | 2 | — | |
CYYAXTCZGPRATM
|
6.5 | IC50 | 2 | — | |
FUNHEVBLXUQXLG
|
6.5 | IC50 | 2 | — | |
IYAVTZWBGCXXFI
|
6.5 | IC50 | 2 | — | |
LLVALEUPUXIQNY
|
6.5 | IC50 | 2 | — | |
NDSMOKBIZMIYDJ
|
6.5 | IC50 | 2 | — | |
QOXCLDKXSCBOOF
|
6.5 | IC50 | 3 | — | |
RJAXVZUSTIFVGP
|
6.5 | IC50 | 2 | — | |
RXGPCIHYSMKIRI
|
6.5 | Ki | 2 | — | |
VJVSHXVHOJVSOB
|
6.5 | Ki | 3 | — | |
CTRVTEOXKBMCKO
|
6.5 | IC50 | 3 | — | |
DWDIQEPGVYBABO
|
6.5 | IC50 | 3 | — | |
GUSAOPYZFQQULB
|
6.5 | IC50 | 2 | — | |
HHZIURLSWUIHRB
|
6.5 | IC50 | 57 | Yes | |
RDTDFCZCBIXFEI
|
6.5 | IC50 | 5 | — | |
RFAXDYWZHZWHAW
|
6.5 | IC50 | 2 | — | |
RFAXDYWZHZWHAW
|
6.5 | IC50 | 2 | — | |
WLXLHHAZRRMMDZ
|
6.5 | IC50 | 2 | — | |
CGJVMKJGKFEHTL
|
6.5 | IC50 | 3 | — | |
DIFGSGNUHRNWPK
|
6.5 | IC50 | 5 | — | |
GDSVOHILVQPEJQ
|
6.5 | IC50 | 2 | — | |
GMIVYDCUSUDJGH
|
6.5 | IC50 | 2 | — | |
HAYGNNHVUSBUBN
|
6.5 | Ki | 3 | — | |
HGBUYZBCPZIMRH
|
6.5 | IC50 | 2 | — | |
HILQSLVIBNFOMC
|
6.5 | IC50 | 2 | — | |
KDARXVILVONBOM
|
6.5 | IC50 | 2 | — | |
LOUPRKONTZGTKE
|
6.5 | IC50 | 2 | — | |
PESOUNLSPHQJGL
|
6.5 | IC50 | 2 | — |