Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZSGUUFCXNQUDKV
|
6.6 | Ki | 2 | — | |
BWBOBCUPLKYBOV
|
6.6 | IC50 | 3 | — | |
CHLHMGGBVMLLOD
|
6.6 | IC50 | 2 | — | |
PCAMVFAVWHIYLC
|
6.6 | IC50 | 2 | — | |
VILNAIPEYFWQQH
|
6.6 | IC50 | 2 | — | |
GXIFPPFQXPIEKY
|
6.6 | Ki | 2 | — | |
IKMISGUCMXQLNN
|
6.6 | Ki | 2 | — | |
JCSQJXFZDFSQLX
|
6.6 | IC50 | 2 | — | |
MNJPFSBAYJQZOE
|
6.6 | IC50 | 3 | — | |
WWYCEUZRECUBAR
|
6.6 | Ki | 2 | — | |
ZQADELCMZHYIPT
|
6.6 | IC50 | 2 | — | |
UGRYBQQJOKDQHB
|
6.6 | IC50 | 2 | — | |
ZMOPTLXEYOVARP
|
6.6 | IC50 | 14 | Yes | |
AWCUGJTVKPBYHS
|
6.6 | IC50 | 2 | — | |
AZIHSCHAYYVWIY
|
6.6 | IC50 | 2 | — | |
BDJJZYXDJQVPIV
|
6.6 | IC50 | 2 | — | |
CNNSTIWPQJEDBI
|
6.6 | IC50 | 3 | — | |
DRKUAUJUSZGTGW
|
6.6 | IC50 | 3 | — | |
FBOUYBDGKBSUES
|
6.6 | IC50 | 6 | — | |
GOKWVWMOVLFRQZ
|
6.6 | IC50 | 2 | — | |
GPRHHSZIXIDKDN
|
6.6 | IC50 | 3 | — | |
INZVCQWDAXDGMY
|
6.6 | IC50 | 3 | — | |
IYZBRQAAJGEDNI
|
6.6 | IC50 | 3 | — | |
JPVGYGPMNFNVTR
|
6.6 | Ki | 2 | — | |
KEOZDNQHXGUGES
|
6.6 | IC50 | 2 | — | |
KMFDXNUGIFDFHQ
|
6.6 | IC50 | 5 | — | |
LJDQESSYTJNKOI
|
6.6 | IC50 | 2 | — | |
MJLHCRFMFPSGBF
|
6.6 | IC50 | 2 | — | |
MYIVBWHBNPYKLU
|
6.6 | IC50 | 3 | — | |
NAFIXABLSKOHPB
|
6.6 | IC50 | 2 | — | |
OSYDLANVDZCPRE
|
6.6 | IC50 | 3 | — | |
PMOFOATUAABMTD
|
6.6 | IC50 | 2 | — | |
PZBTVBSLNQDOCG
|
6.6 | IC50 | 2 | — | |
QRWDBCPLADXSGV
|
6.6 | IC50 | 2 | — | |
QWMBVXDLQBRGEQ
|
6.6 | IC50 | 3 | — | |
RGQXJYRGDMABLT
|
6.6 | IC50 | 3 | — | |
RKDBVDKLNHXCIZ
|
6.6 | IC50 | 3 | — | |
STIWHEMFVTWALB
|
6.6 | IC50 | 5 | — | |
SXAROQNHORDUFM
|
6.6 | IC50 | 7 | — | |
UDALZSDRQUNHRU
|
6.6 | IC50 | 4 | — | |
VTGDLGOSPAKXEA
|
6.6 | IC50 | 3 | — | |
VTSMNPQRBXHIOD
|
6.6 | IC50 | 3 | — | |
VUFRFPUOFHXBBM
|
6.6 | IC50 | 2 | — | |
WYPKPMSOWOXCPF
|
6.6 | Ki | 2 | — | |
XFJSBMXXKPHIIX
|
6.6 | Ki | 2 | — | |
XSBNGDJHMKLOOQ
|
6.6 | IC50 | 2 | — | |
YFGUGMIFVSSOJY
|
6.6 | IC50 | 2 | — | |
YJTUMJAALUNJJT
|
6.6 | IC50 | 2 | — | |
ZIQDGXNDXRMRPM
|
6.6 | IC50 | 3 | — | |
ZKVBATRJUREUMS
|
6.6 | IC50 | 2 | — |