Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SCBFPLDUOJGCDI
|
6.7 | IC50 | 2 | — | |
SFVKVHVOODTRCH
|
6.7 | IC50 | 2 | — | |
SFVKVHVOODTRCH
|
6.7 | IC50 | 2 | — | |
SGTNSNPWRIOYBX
|
6.7 | IC50 | 19 | — | |
UDUUCGMSUBUXNS
|
6.7 | IC50 | 3 | — | |
UJLZUVUUHZVHFF
|
6.7 | IC50 | 2 | — | |
UOHXUSCZQJMWQO
|
6.7 | IC50 | 2 | — | |
VGIGHGMPMUCLIQ
|
6.7 | Ki | 12 | — | |
WHBCDNPPOUFKAB
|
6.7 | IC50 | 2 | — | |
WYRUGBCTQBZIHO
|
6.7 | IC50 | 5 | Yes | |
XCFWDLWOCXSJOK
|
6.7 | IC50 | 2 | — | |
XZBYXXDYCMUFTP
|
6.7 | IC50 | 3 | — | |
XZXRXUCWJOQZBL
|
6.7 | IC50 | 3 | — | |
YLRVVUNTBVYUEG
|
6.7 | IC50 | 3 | — | |
ZUXRZVPVHVFNSX
|
6.7 | IC50 | 5 | — | |
ZYQHRABKRQWTBJ
|
6.7 | IC50 | 2 | — | |
BGJXBVUWLFEJNM
|
6.7 | IC50 | 3 | — | |
CQCYZYXYLGEQJN
|
6.7 | IC50 | 2 | — | |
GPSVSZZDAKVKII
|
6.7 | Ki | 2 | — | |
OJFKDXVECGWNTB
|
6.7 | IC50 | 2 | — | |
TXEGIIUTZDNUKA
|
6.7 | IC50 | 3 | — | |
CDOLWFQFQZOXNZ
|
6.7 | IC50 | 2 | — | |
DVQXAHGZSWJSQT
|
6.7 | IC50 | 2 | — | |
FUSKAZYRYKJDCI
|
6.7 | IC50 | 2 | — | |
JFOMYMQQAYLFEE
|
6.7 | IC50 | 2 | — | |
KPLQQMQZQUMPCN
|
6.7 | Ki | 2 | — | |
OBXLXUGOZZWQOW
|
6.7 | IC50 | 2 | — | |
OZXPSVBSQRGYFB
|
6.7 | IC50 | 2 | — | |
WNWBYUIGGUXYAA
|
6.7 | Ki | 2 | — | |
ISXKOYQKBFARFC
|
6.7 | Ki | 3 | — | |
KXJVMFXTTSRQMV
|
6.7 | Ki | 2 | — | |
DZZKIDMXCAMPCD
|
6.7 | IC50 | 2 | — | |
FQBBSOFRGNNFDV
|
6.7 | Ki | 3 | — | |
HHCUIUUICDIYLM
|
6.7 | IC50 | 2 | — | |
LLMDFLGIOTWWTF
|
6.7 | IC50 | 2 | — | |
MSOUIIHPMJCUNI
|
6.7 | IC50 | 4 | — | |
OMUJKTRTLSRKRV
|
6.7 | IC50 | 2 | — | |
SGDWPIDXMHBDQC
|
6.7 | IC50 | 4 | — | |
ZLIAFORUHVKWQY
|
6.7 | IC50 | 2 | — | |
DWDIQEPGVYBABO
|
6.7 | IC50 | 3 | — | |
HZISGJVOPZSKRZ
|
6.7 | IC50 | 3 | — | |
NCJKKRRMGQPBBA
|
6.7 | IC50 | 2 | — | |
SORMGDAGOZUFDS
|
6.7 | Ki | 3 | — | |
UICYMQZXHRACIG
|
6.7 | Ki | 2 | — | |
NRNPLYWFPSCQAF
|
6.6 | IC50 | 3 | — | |
OUVWZPPMRFXVAK
|
6.6 | IC50 | 3 | — | |
WRHXPUBAPLIIDL
|
6.6 | IC50 | 2 | — | |
WXPNDRBBWZMPQG
|
6.6 | IC50 | 28 | — | |
XYXAYUQJAMPEPZ
|
6.6 | IC50 | 2 | — | |
YNNUSGIPVFPVBX
|
6.6 | Ki | 24 | Yes |