Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KVWDHTXUZHCGIO
|
6.7 | IC50 | 32 | Yes | |
MYCSOYFHSBECSR
|
6.7 | IC50 | 2 | — | |
NJNUNXVUFLFRNF
|
6.7 | Ki | 2 | — | |
RNPOMBJFPXUWGB
|
6.7 | IC50 | 3 | — | |
WLEUBRYSZJGDFY
|
6.7 | IC50 | 4 | — | |
BFGRVRCTCWRWNN
|
6.7 | IC50 | 2 | — | |
GVCHBMCBPBRORW
|
6.7 | IC50 | 3 | — | |
KUUYARHPFYBLLJ
|
6.7 | IC50 | 2 | — | |
MJJALKDDGIKVBE
|
6.7 | IC50 | 30 | Yes | |
AAXGNXOJOSOUQQ
|
6.7 | IC50 | 3 | Yes | |
KKKGFVLMGTXNNX
|
6.7 | Ki | 2 | — | |
MNAFRWGRFIBAQX
|
6.7 | IC50 | 4 | — | |
NBVPHNBDESFHFB
|
6.7 | IC50 | 2 | — | |
XBIDNEGDXXMQIB
|
6.7 | Ki | 2 | — | |
YXQCOSKWQAQJJN
|
6.7 | IC50 | 2 | — | |
NDJMUWDIDQMYFY
|
6.7 | Ki | 4 | — | |
OTJQQIAODOJEAU
|
6.7 | IC50 | 2 | — | |
ZAAQJDPTTZJUDL
|
6.7 | Ki | 4 | — | |
AAONJNLMLWRZJE
|
6.7 | IC50 | 3 | — | |
ABJLUTPPUMSFJV
|
6.7 | IC50 | 2 | — | |
ABJLUTPPUMSFJV
|
6.7 | IC50 | 2 | — | |
AKTHZRZKYPJJRC
|
6.7 | Ki | 4 | — | |
AMADCPJVPLUGQO
|
6.7 | IC50 | 2 | — | |
BEPIQXLVCZPKMN
|
6.7 | IC50 | 3 | — | |
BJKBLXBZYXGWIS
|
6.7 | Ki | 2 | — | |
CEJBRQBGHDEPNJ
|
6.7 | IC50 | 4 | — | |
CUOZZEMLTFRECQ
|
6.7 | IC50 | 3 | — | |
DGKURWUVIVQHCD
|
6.7 | Ki | 2 | — | |
DOKSQMPMAHUKLJ
|
6.7 | Ki | 2 | — | |
DOTHXJXYLNKQOQ
|
6.7 | IC50 | 2 | — | |
DPSHYRRSRHVRRE
|
6.7 | Ki | 2 | — | |
GFQPGTMHAHWZHS
|
6.7 | Ki | 4 | — | |
GOLAHDQVVNCLCU
|
6.7 | IC50 | 3 | — | |
GRYXYXQISNGOHR
|
6.7 | IC50 | 3 | — | |
IONCAKHVNMAPQA
|
6.7 | IC50 | 3 | — | |
JMYVVZJJTRVCDC
|
6.7 | Ki | 2 | — | |
KGNWCYQCPGINGS
|
6.7 | IC50 | 4 | — | |
KGUDOEAVFUTLFC
|
6.7 | Ki | 2 | — | |
KXPNLMZWAKJGRB
|
6.7 | IC50 | 2 | — | |
LPOUMFNXXSGLCK
|
6.7 | IC50 | 7 | — | |
MHPHRNFSAZNRAT
|
6.7 | IC50 | 2 | — | |
MSUDNEADKNPNRJ
|
6.7 | IC50 | 2 | — | |
NASKVDWGYKOGBO
|
6.7 | Ki | 2 | — | |
NHJGZNMVTILZTQ
|
6.7 | Ki | 5 | — | |
NWICMXBOJMLOIB
|
6.7 | IC50 | 3 | — | |
OWNUCKLLDLFPLN
|
6.7 | IC50 | 3 | — | |
QYAPJFAWWAJNJA
|
6.7 | IC50 | 3 | — | |
QZEXFNKCPOFGAE
|
6.7 | IC50 | 2 | — | |
RKTWFMDUKBINRA
|
6.7 | Ki | 5 | — | |
RWNXMLKAIWDHLU
|
6.7 | IC50 | 5 | — |