Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AWJOAMPQOUEKCN
|
6.8 | IC50 | 2 | — | |
CIAWHNGOFJZBCL
|
6.8 | IC50 | 5 | — | |
DFEVQPHSPAIFED
|
6.8 | IC50 | 4 | — | |
GIEBQTVDYXTBCS
|
6.8 | Ki | 2 | — | |
IEQYRWPMNVPDLX
|
6.8 | IC50 | 2 | — | |
IHXFHHOZRJEQBX
|
6.8 | IC50 | 2 | — | |
IRCISBCAVGOJIS
|
6.8 | IC50 | 2 | — | |
JCZQORKBTOWEKS
|
6.8 | IC50 | 3 | — | |
KGQCLTUHOICIST
|
6.8 | IC50 | 2 | — | |
MHFKMHGOYNDZEI
|
6.8 | Ki | 2 | — | |
NAGKIWFBALBSMD
|
6.8 | Ki | 2 | — | |
OHAOVJVRDRFORL
|
6.8 | IC50 | 2 | — | |
OUEZWZJJIKBFFV
|
6.8 | IC50 | 5 | — | |
QDLQBKBQLRPJEG
|
6.8 | Ki | 2 | — | |
RIEBHVBGMUWBCP
|
6.8 | IC50 | 4 | — | |
UKPYAHVTVCYHSG
|
6.8 | IC50 | 3 | — | |
VWVVYFJIUBMXBZ
|
6.8 | IC50 | 2 | — | |
XGXDWBUGQKHTSH
|
6.8 | IC50 | 3 | — | |
XHUFNAKJPMHBAE
|
6.8 | Ki | 2 | — | |
YUGLAKINIYKKIY
|
6.8 | IC50 | 3 | — | |
ZLAONGKKHFSBFL
|
6.8 | IC50 | 3 | — | |
FGXWKSZFVQUSTL
|
6.8 | IC50 | 10 | Yes | |
GMJXFEMNNKZIHB
|
6.8 | Ki | 4 | — | |
RAPZEAPATHNIPO
|
6.8 | IC50 | 28 | Yes | |
VWZIWKHACUENGU
|
6.8 | IC50 | 2 | — | |
ODSCFSVBFVSJFO
|
6.8 | IC50 | 2 | — | |
PHDDUIXSXSRRQU
|
6.8 | Ki | 4 | — | |
SUAKAXXIPDSKLQ
|
6.8 | IC50 | 2 | — | |
HKUKEMRCCWWBFD
|
6.8 | IC50 | 2 | — | |
JXONLPOCIBGKJY
|
6.8 | Ki | 2 | — | |
KYCOIXNLEBVXEA
|
6.8 | IC50 | 2 | — | |
UYLZHMAXLJBXOB
|
6.8 | IC50 | 2 | — | |
XPHJICKYBJRKLW
|
6.8 | IC50 | 2 | — | |
YOQCIOKHHDUPPQ
|
6.8 | IC50 | 2 | — | |
IYIKLHRQXLHMJQ
|
6.8 | IC50 | 18 | — | |
JCCNYMKQOSZNPW
|
6.8 | IC50 | 4 | — | |
KJPJMTVTIDGCRM
|
6.8 | IC50 | 2 | — | |
XKPVANIUEZWDCZ
|
6.8 | IC50 | 2 | — | |
DLEHGKOYLBSEGL
|
6.8 | IC50 | 2 | — | |
DUAKQKCVTZFHSD
|
6.8 | IC50 | 2 | — | |
GZCPBKYTXSPNQJ
|
6.8 | IC50 | 2 | — | |
JGAPWJRMEQDHGG
|
6.8 | IC50 | 2 | — | |
KYCWFOMNQICMSP
|
6.8 | Ki | 2 | — | |
VINPUJZJRCEBET
|
6.8 | IC50 | 5 | — | |
BNPYZAAZLNWAPS
|
6.7 | Ki | 3 | — | |
FMNHTBXXYZCSCU
|
6.7 | IC50 | 4 | — | |
GKIRPKYJQBWNGO
|
6.7 | IC50 | 4 | — | |
GLYFGYIXZOBFGF
|
6.7 | Ki | 2 | — | |
HSHBIVVLOXFRND
|
6.7 | IC50 | 2 | — | |
KLQBJPKPQBLAOR
|
6.7 | IC50 | 2 | — |