Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CLYZVNJXJPXTED
|
6.9 | IC50 | 3 | — | |
DSJQIICDRFEFMZ
|
6.9 | IC50 | 3 | — | |
FLIIXHVRMXEDPQ
|
6.9 | IC50 | 3 | — | |
IZZNYYLQSUDWDO
|
6.9 | IC50 | 3 | — | |
MVWVFYHBGMAFLY
|
6.9 | IC50 | 31 | Yes | |
RPAZQDWESIXCRX
|
6.9 | IC50 | 3 | — | |
SQQYHALTXOFUNG
|
6.9 | IC50 | 3 | — | |
VUFRFPUOFHXBBM
|
6.9 | IC50 | 2 | — | |
AECDBHGVIIRMOI
|
6.9 | IC50 | 7 | — | |
BTEHVLUMUBTQOZ
|
6.9 | IC50 | 3 | — | |
GLVRFLRDWCHDAD
|
6.9 | IC50 | 2 | — | |
GUGOEEXESWIERI
|
6.9 | IC50 | 18 | Yes | |
ONJYCUBPRIPKCO
|
6.9 | IC50 | 2 | — | |
QVIIMXQIBJRPFS
|
6.9 | IC50 | 3 | — | |
VAKGFJFMMQQEIE
|
6.9 | IC50 | 2 | — | |
VHSIEYYFBUUDJV
|
6.9 | Ki | 2 | — | |
WPBRSJXCRWSAHJ
|
6.9 | IC50 | 2 | — | |
YDNXGTGGTKAMFI
|
6.9 | IC50 | 2 | — | |
ZSXSCBZZKDDDST
|
6.9 | IC50 | 3 | — | |
ZTRXHQCTETXYCC
|
6.9 | IC50 | 3 | — | |
KLBQZWRITKRQQV
|
6.9 | IC50 | 21 | — | |
KLQDZSYTMPJBBU
|
6.9 | IC50 | 3 | — | |
PHCUGENQVJPTLC
|
6.9 | Ki | 4 | — | |
VMFNUQHBZCMQRZ
|
6.9 | Ki | 2 | — | |
VRVONDCSZOZMRU
|
6.9 | IC50 | 2 | — | |
LSIUKLXQSPBSEE
|
6.9 | Ki | 3 | — | |
ZQXPNWSXFWKXRZ
|
6.9 | Ki | 2 | — | |
CTNRLCXTSKIWEA
|
6.8 | IC50 | 2 | — | |
TWNPKIQHYYMCGF
|
6.8 | IC50 | 2 | — | |
TXFFWCPTQAOPNJ
|
6.8 | IC50 | 2 | — | |
YIHQDWZWZRGAIH
|
6.8 | IC50 | 9 | — | |
BNJWMFYATZFMQM
|
6.8 | Ki | 2 | — | |
LKIZJVWLCHAZTJ
|
6.8 | IC50 | 3 | — | |
NATFNVDYLPURMJ
|
6.8 | Ki | 4 | — | |
BXUOVUWILQWARZ
|
6.8 | Ki | 3 | — | |
FOBFICSYUINKAA
|
6.8 | IC50 | 6 | — | |
HBGLVJABBICLQC
|
6.8 | Ki | 2 | — | |
HLRRHIITKGDLDO
|
6.8 | Ki | 2 | — | |
IRENZKMIJSGHBF
|
6.8 | IC50 | 3 | — | |
LHFRREYTABIJEO
|
6.8 | Ki | 4 | — | |
LJCOFEDAMMEFHX
|
6.8 | IC50 | 2 | — | |
NCDCQNWXYJMYAZ
|
6.8 | IC50 | 2 | — | |
NIFGQHGFOUMQJN
|
6.8 | IC50 | 5 | — | |
PHCHRPWAMGPRTQ
|
6.8 | Ki | 2 | — | |
PLCSPMWUVPYGEZ
|
6.8 | IC50 | 2 | — | |
QSMZHNDKHVVMTF
|
6.8 | Ki | 2 | — | |
VGTIZFQOKBYTEW
|
6.8 | IC50 | 2 | — | |
VKQSAQSCKUZTCV
|
6.8 | IC50 | 3 | — | |
APXWTOJVYSVWJO
|
6.8 | IC50 | 2 | — | |
ARXBAOIZXCCQAV
|
6.8 | IC50 | 3 | — |