Target Details
| UniProt AC | Q12809 |
|---|---|
| Gene Symbol | KCNH2 |
| Protein Name | Voltage-gated inwardly rectifying potassium channel KCNH2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00027 (cNMP_binding) PF00520 (Ion_trans) PF13426 (PAS_9) |
Summary
- Multi-target molecules 1,607
- Clinical molecules 36
- Avg pChEMBL 6.75
Associated Diseases (2)
Active Molecules (1,607)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZFHQLTFHZHQXAS
|
10.7 | IC50 | 4 | — | |
NBCIMSDAMDKCQO
|
9.8 | IC50 | 3 | — | |
VAXBZBVXSWAUTJ
|
9.8 | IC50 | 2 | — | |
XWQQRPSPOBDJLI
|
9.8 | IC50 | 40 | — | |
GIEKCIRAZIHHMU
|
9.6 | IC50 | 3 | — | |
RLHOWHVHHMGIKE
|
9.6 | IC50 | 3 | — | |
LWMPULARVSIYHV
|
9.4 | IC50 | 3 | — | |
KNKVLWDIKQGTIB
|
9.4 | IC50 | 2 | — | |
BFTJQHWCWUZADH
|
9.3 | IC50 | 2 | — | |
IQNJFMKUOZAASF
|
9.2 | IC50 | 2 | — | |
ITIBCQXWZIYCDK
|
9.2 | IC50 | 3 | — | |
NBLFFMILGMAYPO
|
9.2 | IC50 | 2 | — | |
OLOYPXPKAJGIQP
|
9.2 | IC50 | 2 | — | |
ZMANQSXBZZYBCV
|
9.2 | IC50 | 2 | — | |
ACZXUEYRPYGYKP
|
9.1 | IC50 | 3 | — | |
IQWBKNWLBVZZLG
|
9.1 | Ki | 2 | — | |
AOWSHKSCOCMIOV
|
9.1 | IC50 | 2 | — | |
MGBCOVVRZAHNAM
|
9.1 | IC50 | 2 | — | |
RDIWNJDCZLGDOS
|
9.1 | IC50 | 2 | — | |
KPNMZYDKYZNYIC
|
9.0 | IC50 | 2 | — | |
GJWFUGSRILNJBR
|
9.0 | IC50 | 4 | — | |
YMJIAMCWLDWKKQ
|
9.0 | IC50 | 2 | — | |
HKOWUXNNUVZKQN
|
9.0 | IC50 | 3 | — | |
XMAQSYOMAMZVAK
|
8.9 | IC50 | 2 | — | |
ZITSWKKGCZZGDB
|
8.9 | IC50 | 2 | — | |
MOSUHPUFLYLQDT
|
8.9 | IC50 | 2 | — | |
OTYQXOHDRTWMJY
|
8.9 | Ki | 2 | — | |
GJWFUGSRILNJBR
|
8.8 | IC50 | 4 | — | |
JFLDPXNTPNHXDV
|
8.8 | IC50 | 2 | — | |
NFWRERNMTFKQTQ
|
8.8 | IC50 | 3 | — | |
XFDBWZWHJOLNAF
|
8.8 | IC50 | 2 | — | |
HJSOKBFUMBEYNW
|
8.8 | IC50 | 2 | — | |
JZADUPQYVWWLBA
|
8.8 | IC50 | 2 | — | |
QFMKXHLMZGDSKW
|
8.8 | IC50 | 2 | — | |
CRBIBFLRQNHOTI
|
8.8 | IC50 | 2 | — | |
NZEFYLGMSWSUDH
|
8.8 | IC50 | 4 | — | |
PSBJWNCYYQWCMX
|
8.8 | IC50 | 2 | — | |
YFSPDWGKSWOSRI
|
8.8 | IC50 | 2 | — | |
DJJJSDVUVOIUKR
|
8.8 | IC50 | 3 | — | |
HOWBDMROKCOABA
|
8.8 | IC50 | 7 | — | |
JLBZQGVJKAWCSE
|
8.8 | IC50 | 2 | — | |
HHXTYKXNOKWJQP
|
8.7 | IC50 | 2 | — | |
LSDCVVODSBVDMA
|
8.7 | IC50 | 2 | — | |
LWSWCRMTCQGGDJ
|
8.7 | IC50 | 2 | — | |
WDHOIABIERMLGY
|
8.7 | IC50 | 3 | — | |
GGSBMAVBGZRJPI
|
8.7 | IC50 | 2 | — | |
LBKZCCBZNZAAMS
|
8.7 | IC50 | 2 | — | |
ZKZMTIDHRGLEJP
|
8.7 | IC50 | 2 | — | |
IVBCTFVBWGUGKC
|
8.7 | IC50 | 2 | — | |
JXLYITXDNWJUQB
|
8.7 | IC50 | 2 | — |