Target Details
| UniProt AC | Q10469 |
|---|---|
| Gene Symbol | MGAT2 |
| Protein Name | Alpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05060 (MGAT2) |
Summary
- Multi-target molecules 45
- Clinical molecules 1
- Avg pChEMBL 7.59
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (45)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XVSKYVJHKGLQMZ
|
9.0 | IC50 | 2 | — | |
JQJHRZJLIRYDBY
|
8.7 | IC50 | 2 | — | |
FBBPRPJENPWDPL
|
8.6 | IC50 | 2 | — | |
AGMJOPGTQYKYQI
|
8.5 | IC50 | 2 | — | |
RGDHGNPUKLLPLT
|
8.5 | IC50 | 2 | — | |
RORNAFSJAHYYEW
|
8.4 | IC50 | 2 | — | |
MDMMWSVMDMOFFW
|
8.4 | IC50 | 2 | — | |
FCGICIUXXYBWOA
|
8.3 | IC50 | 2 | — | |
JGMOZJFBAVTQDX
|
8.3 | IC50 | 2 | — | |
QTMPGZCOTIVWFX
|
8.3 | IC50 | 2 | — | |
VFFPVFKSCNJAMO
|
8.3 | IC50 | 2 | — | |
WDLHNOKAVCEXRE
|
8.2 | IC50 | 2 | — | |
APXWBCMMYGRMJI
|
8.2 | IC50 | 3 | — | |
AEMPUAWUDAMJBV
|
8.2 | IC50 | 2 | — | |
VSZRYLHBOKTNBO
|
8.1 | IC50 | 2 | — | |
WWYKHNKFMVELRK
|
8.1 | IC50 | 2 | — | |
LQEYPJWBBIAXMY
|
8.1 | IC50 | 2 | — | |
OLRFZXNKUYOPOO
|
8.0 | IC50 | 2 | — | |
RTEIGMFFNPUILL
|
8.0 | IC50 | 2 | — | |
FBBPRPJENPWDPL
|
8.0 | IC50 | 2 | — | |
UNUKQMOAEMBFBL
|
7.8 | IC50 | 2 | — | |
NNLBWPQNPXPGSO
|
7.6 | IC50 | 3 | — | |
QBHUGPKPNMGAOH
|
7.6 | IC50 | 3 | — | |
JDKJMWFYBKZWNK
|
7.6 | IC50 | 2 | — | |
PAZCANTUHDBJFY
|
7.5 | IC50 | 2 | — | |
JPEMXCVVEWWZTK
|
7.5 | IC50 | 2 | — | |
CQOIVIPBRFSJBE
|
7.4 | IC50 | 2 | — | |
JOVAPGIWTSHPNY
|
7.4 | IC50 | 2 | — | |
NGRPXYWFBXPHAR
|
7.2 | IC50 | 2 | — | |
NFKXWXGBYYQURZ
|
7.2 | IC50 | 2 | — | |
LCFRZBIATSUWDG
|
7.2 | IC50 | 2 | — | |
VHQDXZUUJOXAPJ
|
7.1 | IC50 | 2 | — | |
HINMMPOGDZQMGF
|
7.0 | IC50 | 2 | — | |
YTDRWNDMSGPTFZ
|
6.9 | IC50 | 2 | — | |
NKKYRKMHAMTKLF
|
6.9 | IC50 | 2 | — | |
GSPNLIJIYRHJOM
|
6.8 | IC50 | 2 | — | |
QKRORJZDERERAF
|
6.8 | IC50 | 2 | — | |
JUONYSHFHZDWHI
|
6.6 | IC50 | 2 | — | |
QIXISXYHZPEVNA
|
6.5 | IC50 | 2 | — | |
BWADCEZQHAZYFA
|
6.4 | IC50 | 2 | — | |
VCFIMVZQVDYSSN
|
6.4 | IC50 | 2 | — | |
XYVLITVGCYXABE
|
6.4 | IC50 | 2 | — | |
MGYPXUREAAPVPW
|
6.1 | IC50 | 2 | — | |
QMPLJAUNMPNDSI
|
6.1 | IC50 | 2 | — | |
DFPAKSUCGFBDDF
|
Clinical | TTD_MultiTarget | 2 | Yes |