Target Details
| UniProt AC | Q09470 |
|---|---|
| Gene Symbol | KCNA1 |
| Protein Name | Potassium voltage-gated channel subfamily A member 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02214 (BTB_2) PF00520 (Ion_trans) |
Summary
- Multi-target molecules 130
- Clinical molecules 0
- Avg pChEMBL 10.69
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NRITUABLUPPUBX
|
10.3 | IC50 | 2 | — | |
ZQSYZKYEPKGXSL
|
10.3 | IC50 | 2 | — | |
MGMJUYGWHGCTJI
|
10.3 | IC50 | 2 | — | |
MMXFZICQTOIBAR
|
10.2 | IC50 | 2 | — | |
HWOSZLZJQKYXHL
|
10.1 | IC50 | 2 | — | |
XWQQRPSPOBDJLI
|
9.8 | IC50 | 40 | — | |
QOGZMGDNFLQOLD
|
9.8 | IC50 | 2 | — | |
IUXTUGDAYSHYDJ
|
9.7 | IC50 | 2 | — | |
UNAHIVOXFACQGW
|
9.6 | IC50 | 2 | — | |
JMGJFYAGKIZLOT
|
9.5 | IC50 | 2 | — | |
HXWRRTCVHCEFEO
|
9.5 | IC50 | 2 | — | |
KWIHOEXEWRNRMW
|
9.3 | IC50 | 2 | — | |
PTSSFSTYSLYKSC
|
9.3 | IC50 | 2 | — | |
MJVNYZRDRDGSII
|
9.2 | IC50 | 2 | — | |
ZUXFPRXJKMTJBL
|
9.2 | IC50 | 2 | — | |
XDSROBYJXCIUIC
|
9.1 | IC50 | 2 | — | |
FCNHGNSESJZBMO
|
9.1 | IC50 | 2 | — | |
PFWOJTLVNOZSGQ
|
9.1 | IC50 | 2 | — | |
IOXBFRBDDWONMY
|
9.0 | IC50 | 2 | — | |
OKHJMRQSVKWXRA
|
8.9 | IC50 | 2 | — | |
AAVNWPCABSDFAJ
|
8.7 | IC50 | 2 | — | |
YRMNNNMNSFWNIR
|
8.6 | IC50 | 2 | — | |
NIJMVPXQBCUKPQ
|
8.5 | IC50 | 2 | — | |
NUCQMWUHUMQXKP
|
8.5 | IC50 | 2 | — | |
XJUAALLCFLCXOY
|
8.0 | IC50 | 2 | — | |
YTMOJRFDMQVJGK
|
7.9 | IC50 | 2 | — | |
VVHJIAHVQAXXRH
|
7.5 | IC50 | 2 | — | |
AWQSFBWLDFPCKC
|
6.9 | IC50 | 3 | — | |
KINMYBBFQRSVLL
|
6.6 | IC50 | 6 | — | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — |