Target Details
| UniProt AC | Q09470 |
|---|---|
| Gene Symbol | KCNA1 |
| Protein Name | Potassium voltage-gated channel subfamily A member 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02214 (BTB_2) PF00520 (Ion_trans) |
Summary
- Multi-target molecules 130
- Clinical molecules 0
- Avg pChEMBL 10.69
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VNGREVHCNCHCJQ
|
11.3 | IC50 | 2 | — | |
XVWQLPOVTHTSFJ
|
11.3 | IC50 | 2 | — | |
XZWJCUBBBUYBFD
|
11.3 | IC50 | 2 | — | |
FGRXJZGFNVYRRD
|
11.2 | IC50 | 2 | — | |
GMLMUPKJSZDJPT
|
11.2 | IC50 | 2 | — | |
GWTGRBPCEXNTCG
|
11.2 | IC50 | 2 | — | |
JNICAHXZNOPBGR
|
11.2 | IC50 | 2 | — | |
MTAPHMRNVNWFCB
|
11.2 | IC50 | 2 | — | |
UFSKNTWMVQIQFI
|
11.2 | IC50 | 2 | — | |
FAYQTGPPHXVFLJ
|
11.2 | IC50 | 2 | — | |
KOSCUQHNZXBJTN
|
11.2 | IC50 | 2 | — | |
WILILEKJWLRYGJ
|
11.2 | IC50 | 2 | — | |
YUWLUQFZKRMTDE
|
11.2 | IC50 | 2 | — | |
CJZCBLZAYLXLEB
|
11.1 | IC50 | 2 | — | |
CLPWVUISSPKSEM
|
11.1 | IC50 | 2 | — | |
DDVDSQYLDSBAJW
|
11.1 | IC50 | 2 | — | |
MCVPVAVCCDIYKZ
|
11.1 | IC50 | 2 | — | |
MDNGTLCZVMBCLY
|
11.1 | IC50 | 2 | — | |
NCFJHDRGQOGCBE
|
11.1 | IC50 | 2 | — | |
ORCJROBPAVLWCS
|
11.1 | IC50 | 2 | — | |
OYMSRNHAWCYXGW
|
11.1 | IC50 | 2 | — | |
AIUQAYTYZVNJRO
|
11.0 | IC50 | 2 | — | |
RAQREEQITKQRCO
|
11.0 | IC50 | 2 | — | |
BJZYXUKLPMRGGH
|
11.0 | IC50 | 2 | — | |
CKPYVPWYQDUZOT
|
11.0 | IC50 | 2 | — | |
QZUMGINDDCDSBP
|
11.0 | IC50 | 2 | — | |
IEGDVJDHRFSJAC
|
10.8 | IC50 | 2 | — | |
BCAVQHJGLXITPN
|
10.8 | IC50 | 2 | — | |
VGPBQBJQLLMKNZ
|
10.8 | IC50 | 2 | — | |
XSSVGYVSNAGLBL
|
10.8 | IC50 | 2 | — | |
LJTSSXVJDHQUSV
|
10.8 | IC50 | 2 | — | |
ISGYCGPNHNCKMX
|
10.7 | IC50 | 2 | — | |
XOYHXUGSOFKYHW
|
10.7 | IC50 | 2 | — | |
GVRGDWHECZKHIP
|
10.7 | IC50 | 2 | — | |
MPJOUXWVQCCQNJ
|
10.7 | IC50 | 2 | — | |
XSNNIJZCKAVDAK
|
10.7 | IC50 | 2 | — | |
WURLFZYSKBPESL
|
10.6 | IC50 | 2 | — | |
NSQPUHWCJPLGPR
|
10.6 | IC50 | 2 | — | |
OOUWDISFEFEHIW
|
10.6 | IC50 | 2 | — | |
VVYWFZMUNLNUCN
|
10.6 | IC50 | 2 | — | |
YMGSFPHRPRBAFF
|
10.6 | IC50 | 2 | — | |
LNILZCFUNKQKGB
|
10.5 | IC50 | 2 | — | |
PDVMTOIBVXVEMS
|
10.5 | IC50 | 2 | — | |
WBCRUAYGKPHAFU
|
10.5 | IC50 | 2 | — | |
OKQRSTUYZADHIM
|
10.5 | IC50 | 2 | — | |
GSILMIYKRCUJFS
|
10.4 | IC50 | 2 | — | |
MNHNQVHNKNMYAI
|
10.4 | IC50 | 2 | — | |
NAWHDDMQVAJNNL
|
10.4 | IC50 | 2 | — | |
QONNQPSPJLMZRQ
|
10.3 | IC50 | 2 | — | |
DCXXBQMGZMBPTB
|
10.3 | IC50 | 2 | — |