Target Details
| UniProt AC | Q09470 |
|---|---|
| Gene Symbol | KCNA1 |
| Protein Name | Potassium voltage-gated channel subfamily A member 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02214 (BTB_2) PF00520 (Ion_trans) |
Summary
- Multi-target molecules 130
- Clinical molecules 0
- Avg pChEMBL 10.69
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (130)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DLAPEPHYVMGKDA
|
12.0 | IC50 | 2 | — | |
ISHQEKHPGJKAOO
|
12.0 | IC50 | 2 | — | |
JUIHQJSEZIKHIB
|
12.0 | IC50 | 2 | — | |
QIPIGJQKZYTJRZ
|
12.0 | IC50 | 2 | — | |
XOIPSZFYZUODPP
|
12.0 | IC50 | 2 | — | |
AXPILTLUBXWORL
|
11.7 | IC50 | 2 | — | |
CLLKDYXUEDEDPR
|
11.7 | IC50 | 2 | — | |
CSBUODFTALORPJ
|
11.7 | IC50 | 2 | — | |
GGOFNRIKKIHBMH
|
11.7 | IC50 | 2 | — | |
GTVIZXWFXNFJFH
|
11.7 | IC50 | 2 | — | |
IETAKUSAVBPBNG
|
11.7 | IC50 | 2 | — | |
OLZRHVFWMXZNMK
|
11.7 | IC50 | 2 | — | |
ROADZYRBNDCTEU
|
11.7 | IC50 | 2 | — | |
XBEOCUXEKFHXDW
|
11.7 | IC50 | 2 | — | |
XLIJKTNAZVSZOH
|
11.7 | IC50 | 2 | — | |
YYFOLISOLSRUEH
|
11.7 | IC50 | 2 | — | |
CLYBEGAYCADINR
|
11.5 | IC50 | 2 | — | |
CVJDNZMRVZDVMI
|
11.5 | IC50 | 2 | — | |
DZKBIQQHQXVCLG
|
11.5 | IC50 | 2 | — | |
FCXTYHBPHIJONH
|
11.5 | IC50 | 2 | — | |
FGIIXYFGJJQSRB
|
11.5 | IC50 | 2 | — | |
JUNDLAPHTHBRCO
|
11.5 | IC50 | 2 | — | |
JZIARQXHYOZLDB
|
11.5 | IC50 | 2 | — | |
OLXBZSNTKWJMPP
|
11.5 | IC50 | 2 | — | |
QERLZWREKHBWBR
|
11.5 | IC50 | 2 | — | |
RGLNQBQFWJRABU
|
11.5 | IC50 | 2 | — | |
VSMRVDFLWXBTCO
|
11.5 | IC50 | 2 | — | |
WOGDGDMYCAFOCY
|
11.5 | IC50 | 2 | — | |
XSYVFCNZDMRQTM
|
11.5 | IC50 | 2 | — | |
AEHZNVJYHXWYNR
|
11.4 | IC50 | 2 | — | |
AKYAMZCAYBDMOW
|
11.4 | IC50 | 2 | — | |
BCPMPYAPSPQFAT
|
11.4 | IC50 | 2 | — | |
DKWPCIWMIFPJAZ
|
11.4 | IC50 | 2 | — | |
FURVYTLUPQTUFT
|
11.4 | IC50 | 2 | — | |
GJEQUWMGUKXCSR
|
11.4 | IC50 | 2 | — | |
JZGNOGAGEAKQMK
|
11.4 | IC50 | 2 | — | |
KGCRYMMETKULEM
|
11.4 | IC50 | 2 | — | |
PBQAFRYWKSMSLJ
|
11.4 | IC50 | 2 | — | |
VTRSUFSXBGKQLT
|
11.4 | IC50 | 2 | — | |
VZNSNINLUPDFHE
|
11.4 | IC50 | 2 | — | |
YWLKOPSCCAGKKB
|
11.4 | IC50 | 2 | — | |
ZSCUCOXCDWPNMY
|
11.4 | IC50 | 2 | — | |
AMVJLWLQSQKMFM
|
11.3 | IC50 | 2 | — | |
GZMJRCVVJQKSDM
|
11.3 | IC50 | 2 | — | |
OVQPOMHBBAFOQK
|
11.3 | IC50 | 2 | — | |
OXMAPZLADZSWCZ
|
11.3 | IC50 | 2 | — | |
PKRWQKKLJGZRCR
|
11.3 | IC50 | 2 | — | |
SPXOUPDUGWBDLT
|
11.3 | IC50 | 2 | — | |
SUNRCNJXLTVWOT
|
11.3 | IC50 | 2 | — | |
UNSSOSSHNBBFDP
|
11.3 | IC50 | 2 | — |