Target Details
| UniProt AC | Q09013 |
|---|---|
| Gene Symbol | DMPK |
| Protein Name | Myotonin-protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08826 (DMPK_coil) PF00069 (Pkinase) |
Summary
- Multi-target molecules 20
- Clinical molecules 7
- Avg pChEMBL 6.78
Associated Diseases (1)
Active Molecules (20)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.5 | Kd | 213 | — | |
OATHVDKMFZZHHN
|
7.5 | Kd | 9 | — | |
GDVRVPIXWXOKQO
|
7.5 | IC50 | 10 | — | |
WVUNYSQLFKLYNI
|
7.2 | Kd | 46 | Yes | |
WLKJMISWXHORCR
|
7.2 | IC50 | 11 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
BPNUQXPIQBZCMR
|
7.0 | Kd | 83 | Yes | |
UBPYILGKFZZVDX
|
7.0 | Kd | 130 | Yes | |
OSVUGUHRKMMBSE
|
7.0 | Kd | 170 | — | |
HKSZLNNOFSGOKW
|
7.0 | IC50 | 408 | — | |
MFAQYJIYDMLAIM
|
6.8 | Kd | 130 | Yes | |
UIARLYUEJFELEN
|
6.6 | Kd | 289 | Yes | |
ZCBUQCWBWNUWSU
|
6.5 | Kd | 59 | — | |
JRNJNYBQQYBCLE
|
6.2 | Kd | 40 | Yes | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 82 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JOOXLOJCABQBSG
|
6.0 | Kd | 139 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |