Target Details
| UniProt AC | Q08881 |
|---|---|
| Gene Symbol | ITK |
| Protein Name | Tyrosine-protein kinase ITK/TSK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 676
- Clinical molecules 27
- Avg pChEMBL 7.57
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ILVXQPRFMVXZRH
|
7.6 | IC50 | 2 | — | |
IUPOUNFOIQBJFD
|
7.6 | IC50 | 2 | — | |
MCCCQFAOMZMZKE
|
7.6 | Ki | 52 | — | |
QOSKBOUKENYWAA
|
7.6 | Ki | 2 | — | |
VTZYTGJXYUKXQU
|
7.6 | IC50 | 2 | — | |
VWVYILCFSYNJHF
|
7.6 | Ki | 49 | — | |
WINHZLLDWRZWRT
|
7.6 | Ki | 66 | — | |
FTMHKFYFKGDOSY
|
7.6 | IC50 | 3 | — | |
IZIBDTDSPVBIEA
|
7.6 | IC50 | 2 | — | |
RCDQXYOSLXRXQP
|
7.6 | IC50 | 4 | — | |
CFAYMFXAARPSEQ
|
7.6 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
7.6 | IC50 | 82 | — | |
QNABDSWBQJKBHK
|
7.6 | IC50 | 45 | — | |
YCPPFUIKNAOWRT
|
7.6 | IC50 | 3 | — | |
CBRJPFGIXUFMTM
|
7.6 | Ki | 7 | — | |
RMAUIYTVKFMOGP
|
7.6 | IC50 | 2 | — | |
RMAUIYTVKFMOGP
|
7.6 | IC50 | 2 | — | |
WQFCZTFEEFAYIY
|
7.6 | Ki | 5 | Yes | |
PGXXNNIGDDGRPV
|
7.5 | IC50 | 2 | — | |
DKCAHMDAWGVHSL
|
7.5 | Kd | 3 | — | |
VXUZVATZVGRSHS
|
7.5 | Ki | 2 | — | |
XLCLAYHYRNUKMD
|
7.5 | IC50 | 2 | — | |
KNARVZUUCLIBGV
|
7.5 | Ki | 33 | — | |
XJSFDMGICAWQFS
|
7.5 | Ki | 60 | — | |
ZRFYITKWKPSVFW
|
7.5 | IC50 | 2 | — | |
AQMRYTCSVWYPPS
|
7.5 | IC50 | 2 | — | |
BSJCYMKJSNJNJF
|
7.5 | IC50 | 2 | — | |
BTUKQVNRDONJAO
|
7.5 | IC50 | 2 | — | |
BVGQRQFYDJKNLY
|
7.5 | IC50 | 2 | — | |
CNKBQTIZCNURMG
|
7.5 | IC50 | 2 | — | |
CWTDXPGIFUBVKO
|
7.5 | IC50 | 2 | — | |
DZAHHFCGFLVKIL
|
7.5 | IC50 | 2 | — | |
FBMQVTKLCHHJLB
|
7.5 | IC50 | 2 | — | |
FFYPNJOCHRXBDA
|
7.5 | IC50 | 2 | — | |
GBUXKROHQAKMOJ
|
7.5 | IC50 | 2 | — | |
GNIWWRYROYEXHL
|
7.5 | IC50 | 2 | — | |
GOTJFKXGCMRPAE
|
7.5 | IC50 | 2 | — | |
GSFPDICSPWRBBE
|
7.5 | IC50 | 2 | — | |
HBWIVNIJPLFQBT
|
7.5 | IC50 | 2 | — | |
HGYNVDCJVKJFNP
|
7.5 | IC50 | 2 | — | |
HTZTVRHZAGIUSQ
|
7.5 | IC50 | 2 | — | |
HUBFPPMICSBHGU
|
7.5 | IC50 | 2 | — | |
HUFYIJJOYHBFHQ
|
7.5 | IC50 | 2 | — | |
HZXFVDJXOKIZTO
|
7.5 | IC50 | 2 | — | |
IEVQOCMRVHKNMW
|
7.5 | IC50 | 2 | — | |
IIVMYNDXTSFVTC
|
7.5 | IC50 | 2 | — | |
ILNVUJKWHWBGTL
|
7.5 | IC50 | 2 | — | |
INOPDXCHKQTDEC
|
7.5 | IC50 | 2 | — | |
LJXVSFRUMNKAHQ
|
7.5 | IC50 | 2 | — | |
OARKMUVEVDRZIJ
|
7.5 | IC50 | 2 | — |