Target Details
| UniProt AC | Q08881 |
|---|---|
| Gene Symbol | ITK |
| Protein Name | Tyrosine-protein kinase ITK/TSK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00779 (BTK) PF00169 (PH) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 676
- Clinical molecules 27
- Avg pChEMBL 7.57
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (676)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PWTZWYZDFORBCV
|
9.0 | IC50 | 2 | — | |
STTWMUJSAKOTEV
|
9.0 | IC50 | 4 | — | |
SUHPRCQYTXOSRF
|
9.0 | IC50 | 4 | — | |
CWBFGXHQESGYOA
|
9.0 | IC50 | 4 | — | |
DFNGRDVXGRSFSL
|
9.0 | IC50 | 2 | — | |
YWBAOBYDVWSCMN
|
9.0 | IC50 | 4 | — | |
BQFHXEUTDPRCLM
|
9.0 | IC50 | 4 | — | |
FQYPYAFBYPJBLZ
|
9.0 | IC50 | 2 | — | |
OXVXVYNMDOKNGH
|
9.0 | IC50 | 3 | — | |
MOKNRUDQTSPKQC
|
8.9 | IC50 | 3 | — | |
KWLMYZZUWSGKCI
|
8.9 | IC50 | 4 | — | |
QBTKIUOSXLNHIK
|
8.9 | IC50 | 4 | — | |
YEQGARBJDLREPV
|
8.9 | IC50 | 4 | — | |
NFVGAIXPTCGYPB
|
8.9 | IC50 | 2 | — | |
BOXWOAGQDNNJAR
|
8.9 | IC50 | 4 | — | |
BUXSSQZWDXOIAY
|
8.9 | IC50 | 4 | — | |
FHNCSRKSWPZETL
|
8.9 | IC50 | 4 | — | |
KNEKVQSXRQKRBO
|
8.9 | IC50 | 4 | — | |
IZLUBQPWEKVIDI
|
8.9 | IC50 | 5 | — | |
VMQYRLKWZIILQI
|
8.9 | IC50 | 4 | — | |
MLHBMGYXWLXXSQ
|
8.8 | IC50 | 2 | — | |
KORMETUWFBVJKV
|
8.8 | IC50 | 4 | — | |
UNRUSKKHCUBUIG
|
8.8 | IC50 | 4 | — | |
PWBFGGSRGAQQKP
|
8.8 | IC50 | 4 | — | |
WFTDUNFLISNELR
|
8.8 | IC50 | 4 | — | |
GTMDZIKJMWLLBV
|
8.8 | Ki | 3 | — | |
GZDQSSZYDSPMRO
|
8.8 | IC50 | 3 | — | |
MOWYXIYUNCUBBO
|
8.8 | IC50 | 4 | — | |
NCXHAHGMYXETMO
|
8.8 | IC50 | 2 | — | |
UBWXSCATULGCSA
|
8.8 | IC50 | 4 | — | |
BGHWKOZZYSOJOH
|
8.8 | IC50 | 4 | — | |
CRYRQUNNVGZTRP
|
8.8 | IC50 | 4 | — | |
WQIKESWJRYQGPJ
|
8.8 | IC50 | 3 | — | |
IZIBDTDSPVBIEA
|
8.8 | IC50 | 4 | — | |
OZAGVJOYZGRSJN
|
8.8 | IC50 | 4 | — | |
FHSFSZVDXBNGIW
|
8.8 | IC50 | 4 | — | |
FMUGXGTXXNULGS
|
8.7 | IC50 | 4 | — | |
FVSUKLKFSDSIEF
|
8.7 | IC50 | 4 | — | |
MSIACRQJKTVOPV
|
8.7 | IC50 | 4 | — | |
CLAFAHXMXSENJP
|
8.7 | Ki | 3 | — | |
DJGZDTXKQRIOFX
|
8.7 | IC50 | 2 | — | |
KARRXYMCFAILBZ
|
8.7 | IC50 | 2 | — | |
KWVOXKDNAQPLPP
|
8.7 | IC50 | 2 | — | |
LHVUZIHFLUPGOR
|
8.7 | Ki | 3 | — | |
JKTAWSRABQDLCF
|
8.7 | IC50 | 4 | — | |
ZKLWHHZNVMVOLN
|
8.7 | IC50 | 2 | — | |
FHRWBUZVAOTINV
|
8.7 | IC50 | 4 | — | |
IHIHUZCUZXZSPC
|
8.7 | IC50 | 4 | — | |
LFUKUCJDMFHUGZ
|
8.7 | IC50 | 3 | — | |
LLHYIISPPGQGTN
|
8.7 | IC50 | 2 | — |