Target Details
| UniProt AC | Q08493 |
|---|---|
| Gene Symbol | PDE4C |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4C |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,225
- Clinical molecules 3
- Avg pChEMBL 7.4
KEGG Pathways (5)
Active Molecules (1,225)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKQDIKWPKDHRJH
|
8.8 | IC50 | 4 | — | |
ANSXOWFFAFVDLN
|
8.8 | IC50 | 5 | — | |
HLKIKTJQVCVTJG
|
8.8 | IC50 | 4 | — | |
QIGAIOOPCCZYDO
|
8.8 | IC50 | 4 | — | |
RKHSMIVCRGVSAI
|
8.8 | IC50 | 4 | — | |
CABBMCIEXVVIDP
|
8.8 | IC50 | 4 | — | |
QWJORUKKCABZPO
|
8.7 | IC50 | 4 | — | |
DMPHLSBWKJKTKF
|
8.7 | IC50 | 6 | — | |
GAGSQLMTGCAMOG
|
8.7 | IC50 | 3 | — | |
JFCMFEVPHGDYMS
|
8.7 | IC50 | 4 | — | |
KJUXYSPBVYVNHD
|
8.7 | IC50 | 4 | — | |
LYHFGWILWLEVPK
|
8.7 | IC50 | 2 | — | |
OFNKSFVKBAHXFD
|
8.7 | IC50 | 4 | — | |
SLPPCYGGTCSDJX
|
8.7 | IC50 | 4 | — | |
SMWGOZGGMUJHKG
|
8.7 | IC50 | 4 | — | |
MESOMSSOOSHAJX
|
8.7 | IC50 | 4 | — | |
BIUFOQRGPOVIHK
|
8.7 | IC50 | 3 | — | |
IOHIGXZNGBFEFK
|
8.7 | IC50 | 4 | — | |
SGGQQXATQWLMRQ
|
8.7 | IC50 | 4 | — | |
LSCITVBMOOTYOS
|
8.6 | IC50 | 3 | — | |
UHJAPZBOKPPKGD
|
8.6 | IC50 | 4 | — | |
JTGRNMGEASTCHA
|
8.6 | IC50 | 4 | — | |
XEPASQPUIOGOCW
|
8.6 | IC50 | 4 | — | |
CCJARLANHMJLNZ
|
8.6 | IC50 | 4 | — | |
IPBKYRYKTIGBGW
|
8.6 | IC50 | 4 | — | |
LQUSZPOBAPKYNT
|
8.6 | IC50 | 4 | — | |
WGWKCNVFLGOBOV
|
8.6 | IC50 | 4 | — | |
WPQCJAJFAOGVNJ
|
8.6 | IC50 | 6 | — | |
XZJUOKCCPBELOU
|
8.6 | IC50 | 4 | — | |
XRVDXHQYLWXJOB
|
8.6 | IC50 | 4 | — | |
BBTFKAOFCSOZMB
|
8.6 | IC50 | 5 | — | |
HOKIHKLKOZWCRY
|
8.6 | IC50 | 4 | — | |
JCWCKXNSHPKKEK
|
8.5 | IC50 | 4 | — | |
OEADYOMRQYOJAO
|
8.5 | IC50 | 4 | — | |
WYBLCAXPFFVGGM
|
8.5 | IC50 | 3 | — | |
CEMCFBVPQLOBQK
|
8.5 | IC50 | 2 | — | |
GVLQLBNMZUZFAS
|
8.5 | Ki | 4 | — | |
IXQHNBONEVULTL
|
8.5 | IC50 | 4 | — | |
JERXUPDBWDWFCF
|
8.5 | IC50 | 4 | — | |
KODLAJVZSKZXCU
|
8.5 | IC50 | 2 | — | |
LUUUHUYQTLUIDG
|
8.5 | IC50 | 4 | — | |
MKVXMOXXNMSRPT
|
8.5 | IC50 | 2 | — | |
NAMFJWFHAWRNEK
|
8.5 | IC50 | 2 | — | |
QLKYUVIPOPJNTC
|
8.5 | IC50 | 2 | — | |
TVDXHMKAWBDQFP
|
8.5 | IC50 | 2 | — | |
NMGSQEBMRHQDOG
|
8.5 | IC50 | 4 | — | |
RLKUDKVBRRKFID
|
8.5 | IC50 | 4 | — | |
WOVJAODSYBKIRW
|
8.5 | IC50 | 3 | — | |
DZFTVPIHZOONHV
|
8.5 | IC50 | 4 | — | |
UARYJPSKTPGAFA
|
8.5 | IC50 | 4 | — |