Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OTASYYGEHSXRJI
|
6.3 | IC50 | 3 | — | |
YRCHYHRCBXNYNU
|
6.3 | Kd | 13 | — | |
ODVJDNWZXNGTPP
|
6.2 | IC50 | 2 | — | |
ZBAPBONCBJSTRM
|
6.2 | IC50 | 2 | — | |
KUZZBEKSSYRALS
|
6.2 | Ki | 2 | — | |
XCVSRUFAZODOLV
|
6.2 | IC50 | 2 | — | |
IZGJBYFGTKCESG
|
6.2 | IC50 | 2 | — | |
VLHLGKGZZITZHG
|
6.2 | IC50 | 2 | — | |
FLPLUQYHAQLLOY
|
6.2 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.2 | Kd | 200 | — | |
ULQKNUAMMQCNEF
|
6.2 | IC50 | 2 | — | |
MFAQYJIYDMLAIM
|
6.1 | Kd | 130 | Yes | |
BLQYVHBZHAISJM
|
6.1 | Kd | 21 | Yes | |
RHUJXFIGESXCMV
|
6.1 | IC50 | 2 | — | |
AAKJLRGGTJKAMG
|
6.1 | Kd | 50 | Yes | |
ADWGVRCUXBWAOG
|
6.1 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
6.1 | Kd | 33 | Yes | |
RDUGTASIUXDTFQ
|
6.1 | IC50 | 2 | — | |
JUUFLLKHNYWHKP
|
6.0 | Kd | 12 | — | |
OSVUGUHRKMMBSE
|
6.0 | Kd | 170 | — | |
XYTHPBVXOPRPDS
|
6.0 | IC50 | 2 | — | |
FOWPPHKUFWRWQD
|
6.0 | IC50 | 2 | — | |
MXJKKURRUZSVPI
|
6.0 | IC50 | 2 | — | |
OOHULJHMTVYQJP
|
6.0 | IC50 | 2 | — | |
COEZGIXDSBZROG
|
6.0 | IC50 | 2 | — | |
CDMGBJANTYXAIV
|
6.0 | Kd | 34 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |