Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PDLXVCFCFYZWGX
|
6.7 | IC50 | 2 | — | |
VAPRWSMRTJIVDQ
|
6.6 | IC50 | 4 | — | |
HIROUMBGSVGRCV
|
6.6 | IC50 | 2 | — | |
WAJTXTQMISPZDI
|
6.6 | Ki | 2 | — | |
KDMADGZAPDHVHE
|
6.6 | IC50 | 6 | — | |
BDKBPQWAYIDGNI
|
6.6 | IC50 | 2 | — | |
RAHBGWKEPAQNFF
|
6.6 | Kd | 26 | — | |
IZYYVUMUUJJUFI
|
6.6 | IC50 | 2 | — | |
XURALSVDCFXBAX
|
6.6 | IC50 | 4 | — | |
YAYXNDDVBWDAHB
|
6.6 | IC50 | 2 | — | |
KKKRKRMVJRHDMG
|
6.6 | Kd | 14 | — | |
VLIQZGMHZVDBQW
|
6.6 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
6.6 | Kd | 92 | — | |
YCOYDOIWSSHVCK
|
6.6 | Kd | 10 | — | |
WRVHLHFAAFKTRQ
|
6.5 | IC50 | 2 | — | |
GXMFPDCIAWSZFR
|
6.5 | IC50 | 5 | — | |
HNWYEMIORZATAZ
|
6.5 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.5 | Kd | 599 | — | |
HMLWDEXMRZLYMS
|
6.5 | IC50 | 2 | — | |
ZERKUAJKTYVSGA
|
6.5 | IC50 | 2 | — | |
GZPJCJKUZPUFAL
|
6.5 | Kd | 4 | — | |
ABFDFDOPULQNHT
|
6.5 | IC50 | 2 | — | |
OOYXCHZXSQAPSG
|
6.5 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
6.5 | Kd | 43 | — | |
PCMIKEZTMZXZMY
|
6.5 | IC50 | 2 | — | |
FNHKPVJBJVTLMP
|
6.5 | Kd | 29 | — | |
RUDJLSWOUHMLOU
|
6.5 | IC50 | 3 | — | |
LNMRSSIMGCDUTP
|
6.4 | Kd | 13 | — | |
PTWTZJRZLBYUHC
|
6.4 | IC50 | 2 | — | |
ZQJVDKODUAHTJI
|
6.4 | IC50 | 2 | — | |
VNWJQJZPFFNAKE
|
6.4 | IC50 | 2 | — | |
OMZCMEYTWSXEPZ
|
6.4 | Kd | 43 | Yes | |
SGKRTMGOTGXOAN
|
6.4 | IC50 | 2 | — | |
FNAHTQRLVWZGGT
|
6.4 | IC50 | 2 | — | |
PHNXBYIDBYOSNK
|
6.4 | IC50 | 2 | — | |
MFFNLJJDBHPNPK
|
6.4 | IC50 | 2 | — | |
HDTCSYZQKDPDHW
|
6.3 | IC50 | 3 | — | |
YRXCHCWQVMQAKG
|
6.3 | IC50 | 2 | — | |
VLIQZGMHZVDBQW
|
6.3 | IC50 | 2 | — | |
FLBNLJLONKAPLR
|
6.3 | Kd | 31 | — | |
INQIIYZNPFFIAO
|
6.3 | IC50 | 2 | — | |
XCVSRUFAZODOLV
|
6.3 | IC50 | 2 | — | |
MXJKKURRUZSVPI
|
6.3 | IC50 | 2 | — | |
FFLJVBPCONQSQW
|
6.3 | IC50 | 8 | — | |
WFSMFTUQBULRQN
|
6.3 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
6.3 | Kd | 112 | — | |
IDLGGIATPYXKFN
|
6.3 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 114 | — | |
UIARLYUEJFELEN
|
6.3 | Kd | 289 | Yes | |
ULQKNUAMMQCNEF
|
6.3 | IC50 | 2 | — |