Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VIVYNGHHCGDRHE
|
7.1 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
QGAZPZGGCFPPIQ
|
7.1 | IC50 | 2 | — | |
DXEOLSCGMKPOSP
|
7.0 | IC50 | 2 | — | |
RFKIMRWCLPYQNL
|
7.0 | IC50 | 2 | — | |
UGPDJIJFANODJH
|
7.0 | IC50 | 12 | — | |
YOOBJJUPLPSYTE
|
7.0 | IC50 | 2 | — | |
AOZPVMOOEJAZGK
|
7.0 | IC50 | 2 | — | |
GZMYLSJUNSCMTD
|
7.0 | IC50 | 4 | — | |
HFQACMCWJYLKKX
|
7.0 | IC50 | 2 | — | |
AOWOZJJGVFTXQU
|
7.0 | IC50 | 2 | — | |
IVUGFMLRJOCGAS
|
7.0 | Kd | 9 | — | |
MMSWJNGRQBXTAK
|
7.0 | IC50 | 2 | — | |
XASNYJJSDRRREO
|
7.0 | IC50 | 2 | — | |
DCBIJCAUUCDMMT
|
6.9 | IC50 | 2 | — | |
DQHVUKLVCBJBLM
|
6.9 | IC50 | 8 | — | |
DXEOLSCGMKPOSP
|
6.9 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
6.9 | Kd | 130 | Yes | |
DKNUPRMJNUQNHR
|
6.9 | Kd | 33 | — | |
DSZLKOXKYRREEO
|
6.9 | IC50 | 10 | — | |
XFHUWXYRCAAZHK
|
6.9 | IC50 | 4 | — | |
RCNBJHLIJNEPLE
|
6.9 | IC50 | 2 | — | |
YOHLRCOPRAVUCJ
|
6.9 | IC50 | 6 | — | |
NIIYHUNRXQLMBG
|
6.9 | IC50 | 6 | — | |
FAYAUAZLLLJJGH
|
6.8 | Kd | 36 | Yes | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
XKFTZKGMDDZMJI
|
6.8 | Kd | 64 | Yes | |
AIWDHNDUIDAYMO
|
6.8 | IC50 | 4 | — | |
XVBSTEJSDUMWMA
|
6.8 | IC50 | 3 | — | |
DTGOSWCCJRXHFQ
|
6.8 | IC50 | 2 | — | |
NCCXRWBQPFJCNV
|
6.8 | IC50 | 2 | — | |
AHTIPVCWOOAWGC
|
6.8 | IC50 | 2 | — | |
WCWUXEGQKLTGDX
|
6.8 | Kd | 22 | Yes | |
ZMFVICCTJZQVDM
|
6.8 | IC50 | 3 | — | |
ZCWXCBKGPJOAFQ
|
6.8 | IC50 | 13 | — | |
NQHGDUGVQSAKOR
|
6.8 | IC50 | 3 | — | |
QHADVLVFMKEIIP
|
6.8 | Kd | 9 | — | |
YLNAPFRQMKNPTD
|
6.8 | Ki | 2 | — | |
KOUDZSRFONTIGH
|
6.7 | IC50 | 2 | — | |
SYWCXDMIXNCMEV
|
6.7 | IC50 | 2 | — | |
SPMVMDHWKHCIDT
|
6.7 | Kd | 30 | — | |
FHUUXVNWKWLIFZ
|
6.7 | IC50 | 2 | — | |
FKYPQUFENSTBCR
|
6.7 | IC50 | 2 | — | |
ONIQOQHATWINJY
|
6.7 | Kd | 25 | — | |
QGKXLHRKUNKGPZ
|
6.7 | IC50 | 2 | — | |
JJORFRRMKVGMOJ
|
6.7 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
6.7 | Kd | 55 | — | |
LJODJUIHONTDMR
|
6.7 | IC50 | 7 | — | |
WGYIFHILSUXKKN
|
6.7 | IC50 | 2 | — | |
NVLGVDSMAYCVRY
|
6.7 | IC50 | 2 | — |