Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YVFSNJNTIVOKAV
|
7.4 | IC50 | 2 | — | |
CKCLTNYJBXCOGM
|
7.4 | IC50 | 2 | — | |
DEVDNVYDNDZDRO
|
7.4 | IC50 | 2 | — | |
HDUGVQFEYURLKF
|
7.4 | Ki | 2 | — | |
XFLAQLCDMJRPFH
|
7.4 | IC50 | 5 | — | |
VTBIPUIGATVNGY
|
7.4 | IC50 | 2 | — | |
YBEMAJSTGUDUQZ
|
7.4 | IC50 | 3 | — | |
HKHQEYYGONFDJK
|
7.3 | IC50 | 2 | — | |
UVQRACPXMGFYMZ
|
7.3 | IC50 | 2 | — | |
WOSKHXYHFSIKNG
|
7.3 | Kd | 24 | — | |
GBSOJTHLVSZFNK
|
7.3 | IC50 | 2 | — | |
PBHDCPWPSOSGGD
|
7.3 | IC50 | 2 | — | |
BCABRBNGPCXUDA
|
7.3 | IC50 | 2 | — | |
NHCXDULQCCCWLO
|
7.3 | IC50 | 3 | — | |
WWIJZOWOWLGRSG
|
7.3 | IC50 | 2 | — | |
XLZOLMVQUKURQX
|
7.3 | IC50 | 2 | — | |
QIYCVICASXFGFF
|
7.3 | IC50 | 2 | — | |
OPEMWSXQLXWPSB
|
7.3 | IC50 | 2 | — | |
SUXGZTYFSUWICV
|
7.3 | IC50 | 2 | — | |
VRQMAABPASPXMW
|
7.2 | Kd | 10 | — | |
CUIHSIWYWATEQL
|
7.2 | Kd | 61 | Yes | |
MPVGZUGXCQEXTM
|
7.2 | Kd | 61 | Yes | |
PFTXFNSHFZLJNT
|
7.2 | IC50 | 17 | — | |
DZHWFANVZCHBGK
|
7.2 | IC50 | 2 | — | |
MGKDUWFEPDLKNZ
|
7.2 | IC50 | 2 | — | |
ORYMWWSJZRCUSV
|
7.2 | IC50 | 7 | — | |
AKCMYWNZFYOKFJ
|
7.2 | IC50 | 2 | — | |
SKDBXDGKLQALIZ
|
7.2 | IC50 | 15 | — | |
TZGXRXHVIFVGCP
|
7.2 | IC50 | 2 | — | |
VWMJHAFYPMOMGF
|
7.2 | Kd | 15 | — | |
CEPHPZHFIJLDAZ
|
7.2 | IC50 | 2 | — | |
PFQKMGZTPAMJKD
|
7.2 | IC50 | 2 | — | |
KVGTWUGUDPNRGC
|
7.2 | IC50 | 6 | — | |
KZJMAYVZYCIFHX
|
7.2 | IC50 | 2 | — | |
NVSACWLSRUGEMJ
|
7.2 | IC50 | 2 | — | |
QHJQBVFNRUEDHB
|
7.2 | IC50 | 2 | — | |
SGKRTMGOTGXOAN
|
7.2 | IC50 | 2 | — | |
DZVQBRGQNWDWIG
|
7.2 | IC50 | 6 | — | |
HXHAJRMTJXHJJZ
|
7.2 | Kd | 52 | Yes | |
APMNFDWEFYEHBD
|
7.2 | IC50 | 2 | — | |
OYONTEXKYJZFHA
|
7.2 | Kd | 69 | Yes | |
GNDBDDNLWIOKDN
|
7.2 | IC50 | 5 | — | |
HVXKQKFEHMGHSL
|
7.1 | Kd | 21 | — | |
UKRJOFUVKHRCMD
|
7.1 | IC50 | 2 | — | |
KVOKGAUQGXOEAL
|
7.1 | IC50 | 2 | — | |
NFZXBQXIWXZUDR
|
7.1 | IC50 | 2 | — | |
CVWXJKQAOSCOAB
|
7.1 | Kd | 35 | — | |
QGAZPZGGCFPPIQ
|
7.1 | IC50 | 2 | — | |
SDOMGHNXSMDPGR
|
7.1 | IC50 | 2 | — | |
USBUDHMXOXUPOI
|
7.1 | IC50 | 2 | — |