Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KTUFNOKKBVMGRW
|
7.7 | Kd | 38 | Yes | |
RZOMPFGUSZPJBC
|
7.7 | IC50 | 3 | — | |
WRMITRKGBHCESG
|
7.7 | IC50 | 2 | — | |
CAWFLWKFZFPVQV
|
7.7 | IC50 | 3 | — | |
YIEKEILDJWQXRB
|
7.7 | IC50 | 4 | — | |
JBODBRVQXUEXLM
|
7.6 | IC50 | 2 | — | |
KVCQTKNUUQOELD
|
7.6 | IC50 | 6 | — | |
WGMNFJAFXXXRLZ
|
7.6 | IC50 | 4 | — | |
CPRPVAAUKYCOPQ
|
7.6 | IC50 | 2 | — | |
REAGUYYHFGPZCI
|
7.6 | IC50 | 2 | — | |
YOBIWCLAYQWPPW
|
7.6 | IC50 | 23 | — | |
XJVJYSCTGJVJFB
|
7.6 | IC50 | 2 | — | |
YXESXLYKZKCWFJ
|
7.6 | IC50 | 2 | — | |
DPUOBXMBTCOPQJ
|
7.6 | IC50 | 2 | — | |
DDPFCUXJEFSBMK
|
7.6 | IC50 | 2 | — | |
BGQOUQWQPRPBKN
|
7.6 | IC50 | 7 | — | |
MOONEVNPHKFNGV
|
7.6 | IC50 | 4 | — | |
OSORXAIKGQTSBW
|
7.6 | IC50 | 2 | — | |
LYBOAPPMESGTAR
|
7.6 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
7.5 | Kd | 109 | Yes | |
REKPKQSBXOYNGI
|
7.5 | IC50 | 2 | — | |
UXEXYURPAPXPSR
|
7.5 | IC50 | 2 | — | |
ZFRVWRQOQJYXCC
|
7.5 | IC50 | 2 | — | |
COPFQQYHJSJTAB
|
7.5 | IC50 | 2 | — | |
KHAWCGQVTPTPEV
|
7.5 | IC50 | 2 | — | |
MMSWJNGRQBXTAK
|
7.5 | IC50 | 2 | — | |
XGAYALCZXPVWQM
|
7.5 | IC50 | 2 | — | |
WJTJZDOMFKCYEA
|
7.5 | Kd | 6 | — | |
HBVBUBAJOLRKQP
|
7.5 | IC50 | 2 | — | |
HHZIURLSWUIHRB
|
7.5 | IC50 | 57 | Yes | |
QHBOCRGDNDMWPF
|
7.5 | IC50 | 2 | — | |
XASNYJJSDRRREO
|
7.5 | IC50 | 2 | — | |
AKWLDQDWZNJYKL
|
7.5 | IC50 | 14 | — | |
APPXQUDJLJXULP
|
7.5 | IC50 | 47 | — | |
FLPLUQYHAQLLOY
|
7.5 | IC50 | 2 | — | |
MFZCBEQXFXXPNC
|
7.5 | IC50 | 2 | — | |
XASNYJJSDRRREO
|
7.5 | IC50 | 2 | — | |
DTAKXSCGKBXZTR
|
7.4 | IC50 | 2 | — | |
KSYODHFUZVOSEM
|
7.4 | IC50 | 2 | — | |
SRTRAJZAXAGMAE
|
7.4 | IC50 | 2 | — | |
FXUBVXGXYWZNJY
|
7.4 | IC50 | 2 | — | |
RRUSGGIRDBKDGI
|
7.4 | IC50 | 2 | — | |
SHTNULLAAVPXRC
|
7.4 | IC50 | 4 | — | |
VNBRGSXVFBYQNN
|
7.4 | Kd | 22 | Yes | |
LIGJIQAEZFSGOU
|
7.4 | IC50 | 2 | — | |
MYBCCXGFAIUUOW
|
7.4 | IC50 | 2 | — | |
RFEWCQAWLXXDQI
|
7.4 | IC50 | 5 | — | |
VUJQGYIVERKNSC
|
7.4 | IC50 | 2 | — | |
RKBYYWVZFBATHQ
|
7.4 | IC50 | 12 | — | |
GBSOJTHLVSZFNK
|
7.4 | IC50 | 2 | — |