Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UGRGTNDQCIYUDE
|
7.9 | IC50 | 3 | — | |
SCNJPRUXBGWNTB
|
7.9 | IC50 | 2 | — | |
SERAEYFDVQXTIX
|
7.9 | IC50 | 2 | — | |
ZHAGZTJIWAFRBI
|
7.9 | IC50 | 3 | — | |
CUDVHEFYRIWYQD
|
7.8 | Kd | 11 | — | |
ZGBAJMQHJDFTQJ
|
7.8 | Kd | 15 | — | |
CKFSGFBIQDUWKV
|
7.8 | IC50 | 5 | — | |
DSKYHEJWWIBREA
|
7.8 | IC50 | 8 | — | |
SBGAHKXLTGCPRN
|
7.8 | IC50 | 4 | — | |
XTFQLAOUVSZDDX
|
7.8 | IC50 | 3 | — | |
YEPVECGOLOSJGA
|
7.8 | IC50 | 2 | — | |
YHVHYWYQEFELOW
|
7.8 | IC50 | 44 | — | |
BXIQSHSRUREBOZ
|
7.8 | IC50 | 3 | — | |
HNBOQIQDXUEERR
|
7.8 | IC50 | 2 | — | |
HTLGYDDHGAGGEE
|
7.8 | IC50 | 2 | — | |
RALKOVHFGYUBAB
|
7.8 | IC50 | 5 | — | |
XQZFAZMTCODCDH
|
7.8 | IC50 | 3 | — | |
SYDKMYUOXNXPAU
|
7.8 | IC50 | 2 | — | |
WHHSWSVEDVSZHP
|
7.8 | IC50 | 2 | — | |
ARCVIRDCNNOJSS
|
7.8 | Ki | 2 | — | |
AUYHJDXKEGVPNX
|
7.8 | Ki | 2 | — | |
BDBXXOAYGWEYFR
|
7.8 | IC50 | 2 | — | |
FKYSRBZUEXVNJW
|
7.8 | IC50 | 2 | — | |
FXEZNFCBNZJTKX
|
7.8 | Ki | 2 | — | |
JEXAMDPQBOIWCJ
|
7.8 | Ki | 2 | — | |
LABDHZIYLNNWCF
|
7.8 | IC50 | 2 | — | |
LGJSFFXKADZTNP
|
7.8 | Ki | 2 | — | |
OWRPCKSLYVXUJS
|
7.8 | Ki | 2 | — | |
PKDCZQAKLPJYFN
|
7.8 | Ki | 2 | — | |
YFKFMRKJGPZRSA
|
7.8 | IC50 | 2 | — | |
LIIIOZYEEVCNLB
|
7.8 | IC50 | 2 | — | |
REKPKQSBXOYNGI
|
7.8 | IC50 | 2 | — | |
VDVSFLZBRCBQIQ
|
7.8 | IC50 | 3 | — | |
COPFQQYHJSJTAB
|
7.7 | IC50 | 2 | — | |
CPRPVAAUKYCOPQ
|
7.7 | IC50 | 2 | — | |
DCSRZWOYUOTSMH
|
7.7 | IC50 | 2 | — | |
VVIMBTCNEFBEEY
|
7.7 | IC50 | 2 | — | |
WSOOEDMRKNRFBS
|
7.7 | IC50 | 2 | — | |
CMJJZRAAQMUAFH
|
7.7 | IC50 | 2 | — | |
HLORIUQAGCRNIE
|
7.7 | IC50 | 3 | — | |
MMSWJNGRQBXTAK
|
7.7 | IC50 | 2 | — | |
XAISWZVJRAFMGB
|
7.7 | IC50 | 2 | — | |
ZPCGUXHVTHLYOP
|
7.7 | IC50 | 2 | — | |
KXMZDGSRSGHMMK
|
7.7 | IC50 | 14 | — | |
PGNPRFGVXQKJFG
|
7.7 | IC50 | 4 | — | |
QCSTWBWDCAMLSP
|
7.7 | IC50 | 2 | — | |
GMHKDZXPTJDOJO
|
7.7 | IC50 | 2 | — | |
HYVLWRNCEBMMRK
|
7.7 | IC50 | 2 | — | |
FLPLUQYHAQLLOY
|
7.7 | IC50 | 2 | — | |
IKENQUDOTQBCJH
|
7.7 | IC50 | 18 | — |