Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DDLPXZXBWGJRGK
|
8.2 | IC50 | 4 | — | |
IFVGNYDOUDEVPK
|
8.2 | IC50 | 3 | — | |
CHYCQBZNTKXHMV
|
8.2 | IC50 | 3 | — | |
GYBZVTMKISJGBF
|
8.2 | IC50 | 3 | — | |
OWEGQACAHYGLOT
|
8.1 | IC50 | 3 | — | |
BPQBMWJXOIQOCG
|
8.1 | IC50 | 3 | — | |
OIANGKGOYKDGQV
|
8.1 | Kd | 10 | — | |
QTBWCSQGBMPECM
|
8.1 | Kd | 21 | Yes | |
YYIDVDRESUYFKM
|
8.1 | IC50 | 3 | — | |
XEKBRFPQVSQWMU
|
8.1 | IC50 | 3 | — | |
IALDYVNFZAPNJV
|
8.1 | IC50 | 11 | — | |
ISFMOWLMGGXLTK
|
8.1 | IC50 | 2 | — | |
IUGBGEUCXVKGQK
|
8.1 | IC50 | 13 | — | |
RIWKVLUOTMXONS
|
8.1 | IC50 | 5 | — | |
WJEOLQLKVOPQFV
|
8.1 | Kd | 24 | — | |
BNRXMSGHPVYSDK
|
8.1 | IC50 | 24 | — | |
CTQCFMSNNVNUQZ
|
8.1 | IC50 | 2 | — | |
MXYXKUBTRKHYAM
|
8.1 | IC50 | 3 | — | |
VSVJBCKLXDHEJV
|
8.1 | IC50 | 6 | — | |
KYENXKDRIQKRJP
|
8.0 | IC50 | 5 | — | |
OTKXMYZOSPIKMY
|
8.0 | IC50 | 3 | — | |
CMJJZRAAQMUAFH
|
8.0 | IC50 | 9 | — | |
GUBJNPWVIUFSTR
|
8.0 | Kd | 103 | — | |
NHHQJBCNYHBUSI
|
8.0 | Kd | 220 | — | |
PHXJVRSECIGDHY
|
8.0 | IC50 | 59 | — | |
ZXPUKEPQYKBOHH
|
8.0 | IC50 | 3 | — | |
DAAOYHIERMVREX
|
8.0 | IC50 | 3 | — | |
NYVPWRKNAAFYQA
|
8.0 | IC50 | 2 | — | |
CNFBVUCODRZQOP
|
8.0 | IC50 | 2 | — | |
DTDFVCJCQKMAKM
|
8.0 | IC50 | 2 | — | |
MIMOHMCANSGXIG
|
8.0 | IC50 | 15 | — | |
WFLPERLYBCBHLO
|
8.0 | IC50 | 2 | — | |
FOYGRDAFTLGYQF
|
8.0 | IC50 | 2 | — | |
UHTHHESEBZOYNR
|
8.0 | Kd | 66 | Yes | |
CTZOFTNYJRGNGO
|
8.0 | IC50 | 3 | — | |
LTQIPTSOJUTHQH
|
7.9 | IC50 | 3 | — | |
QTYVZNNBMDNHJL
|
7.9 | IC50 | 3 | — | |
SAAYRHKJHDIDPH
|
7.9 | IC50 | 3 | — | |
SHPFDGWALWEPGS
|
7.9 | Kd | 35 | — | |
XZXHXSATPCNXJR
|
7.9 | Kd | 165 | Yes | |
UHWZHRQDJOKBQY
|
7.9 | IC50 | 3 | — | |
UMQWPKHTVPGLII
|
7.9 | IC50 | 2 | — | |
BCIITSAFUJGIEG
|
7.9 | IC50 | 3 | — | |
GXDWYOLKTKVBFT
|
7.9 | IC50 | 2 | — | |
TYGZNGFFKJJPJQ
|
7.9 | IC50 | 3 | — | |
MWFIUFYSLJRFQM
|
7.9 | IC50 | 2 | — | |
VNRGGLUPXIJJDG
|
7.9 | IC50 | 2 | — | |
YABJJWZLRMPFSI
|
7.9 | Kd | 34 | — | |
DNMQPIQPJLMWPY
|
7.9 | IC50 | 3 | — | |
DRNRCLNUHIQXOJ
|
7.9 | IC50 | 4 | — |