Target Details
| UniProt AC | Q08345 |
|---|---|
| Gene Symbol | DDR1 |
| Protein Name | Epithelial discoidin domain-containing receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21114 (DDR1-2_DS-like) PF00754 (F5_F8_type_C) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 377
- Clinical molecules 28
- Avg pChEMBL 7.38
Active Molecules (377)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CXQHYVUVSFXTMY
|
9.7 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
9.7 | Kd | 149 | — | |
MPASHPJAIUOWCK
|
9.4 | Kd | 9 | — | |
ODPGGGTTYSGTGO
|
9.2 | Kd | 153 | — | |
MLDQJTXFUGDVEO
|
8.8 | Kd | 85 | Yes | |
XXJWYDDUDKYVKI
|
8.8 | Kd | 52 | — | |
IZKVIUJIUTXIRH
|
8.7 | IC50 | 2 | — | |
UEPXBTCUIIGYCY
|
8.7 | Kd | 6 | — | |
ZBNZXTGUTAYRHI
|
8.7 | Kd | 102 | Yes | |
MVCOAUNKQVWQHZ
|
8.7 | Kd | 54 | Yes | |
FHPTWZJZWOYCKG
|
8.7 | IC50 | 5 | — | |
UPXFBKXBRDBIKU
|
8.7 | IC50 | 3 | — | |
UVMSVIJGLODSFN
|
8.7 | IC50 | 3 | — | |
PSBGROLQRNSAMY
|
8.6 | IC50 | 2 | — | |
AYQXKPMEHPZRKR
|
8.6 | IC50 | 6 | — | |
VAARYSWULJUGST
|
8.6 | Kd | 119 | Yes | |
NFTNUHHJWIJBRN
|
8.6 | IC50 | 3 | — | |
AQSSMEORRLJZLU
|
8.5 | Kd | 34 | Yes | |
YXARVHZXTQVAOP
|
8.5 | IC50 | 11 | — | |
QAHANVZHNDZWSM
|
8.5 | IC50 | 3 | — | |
JCNSIZBVFFVTJE
|
8.5 | IC50 | 3 | — | |
KQOYBUCRLZDLBE
|
8.5 | IC50 | 3 | — | |
VTWWRKFUHCSCEW
|
8.5 | Kd | 19 | — | |
DDPFCUXJEFSBMK
|
8.4 | IC50 | 2 | — | |
CYYRPFWAMVGRGT
|
8.4 | IC50 | 3 | — | |
UDRCHZMTVKQTAE
|
8.4 | IC50 | 3 | — | |
IPXKPFIHNPASKD
|
8.4 | IC50 | 2 | — | |
LQSGDXCDNZWTJN
|
8.4 | IC50 | 17 | — | |
XPQJKJDXIUJKQM
|
8.4 | IC50 | 2 | — | |
RRDDKVJWDOIIFN
|
8.4 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.4 | IC50 | 408 | — | |
YXCVYRQZUTUYKZ
|
8.4 | IC50 | 3 | — | |
QCFZDYFUWADUJV
|
8.4 | IC50 | 3 | — | |
VQQKESJQSNYQOP
|
8.3 | IC50 | 3 | — | |
GUFVTKTWKYLOQP
|
8.3 | IC50 | 7 | — | |
UEHGHDJPDQDZPX
|
8.3 | IC50 | 3 | — | |
UQRCJCNVNUFYDX
|
8.3 | Kd | 27 | — | |
VDPIYNSZQSYYGQ
|
8.3 | IC50 | 5 | — | |
BDDFTQKLPQWOLD
|
8.3 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.3 | IC50 | 213 | — | |
XFLAQLCDMJRPFH
|
8.2 | IC50 | 2 | — | |
ITMMHAMHNWGMLK
|
8.2 | IC50 | 2 | — | |
FLOSOQYXYAJVAG
|
8.2 | IC50 | 2 | — | |
KUTDZECNFUUAHC
|
8.2 | IC50 | 3 | — | |
WRRRUTZYQAQDCB
|
8.2 | IC50 | 3 | — | |
LAXWYKGMTZIWKO
|
8.2 | IC50 | 3 | — | |
RZKBSKVRXHFGJG
|
8.2 | IC50 | 3 | — | |
UYAJMVJVPHCOJN
|
8.2 | IC50 | 3 | — | |
CJXZIWDVXAJFBP
|
8.2 | IC50 | 3 | — | |
CZCBVFVSSWZKPW
|
8.2 | IC50 | 3 | — |