Target Details
| UniProt AC | Q07912 |
|---|---|
| Gene Symbol | TNK2 |
| Protein Name | Activated CDC42 kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09027 (GTPase_binding) PF11555 (Inhibitor_Mig-6) PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) PF14604 (SH3_9) |
Summary
- Multi-target molecules 222
- Clinical molecules 22
- Avg pChEMBL 7.46
Active Molecules (222)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GZBRMTRCRSMBNA
|
6.2 | IC50 | 2 | — | |
JWNPDZNEKVCWMY
|
6.2 | Kd | 57 | Yes | |
KTEIFNKAUNYNJU
|
6.1 | Kd | 114 | — | |
AUDNGNGLLRZLDR
|
6.1 | Ki | 33 | — | |
JZTOUVBEZONDKA
|
6.1 | Ki | 80 | — | |
QCOULMVHIHJKFY
|
6.1 | Ki | 14 | — | |
ZLHFILGSQDJULK
|
6.1 | Ki | 37 | Yes | |
GUBJNPWVIUFSTR
|
6.1 | Kd | 103 | — | |
WVUNYSQLFKLYNI
|
6.0 | Kd | 46 | Yes | |
JZVXAFREQFUEDW
|
6.0 | IC50 | 2 | — | |
ZCCPLJOKGAACRT
|
6.0 | Kd | 599 | — | |
APPXQUDJLJXULP
|
6.0 | IC50 | 47 | — | |
BLQYVHBZHAISJM
|
6.0 | Ki | 54 | — | |
GZAQDFYUURXJSL
|
6.0 | Ki | 8 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NKEUPUJTVALZIK
|
6.0 | Ki | 28 | — | |
OONFNUWBHFSNBT
|
6.0 | Kd | 11 | — | |
PBBRWFOVCUAONR
|
6.0 | Ki | 26 | Yes | |
QLWUDWMYFSWGHK
|
6.0 | Ki | 22 | — | |
ZCCJKVBTHCOISJ
|
6.0 | Ki | 46 | — |